Pharmaceutical Co-crystals, Salts, and Co-amorphous Systems: A novel opportunity of hot-melt extrusion
Published 2020 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Pharmaceutical Co-crystals, Salts, and Co-amorphous Systems: A novel opportunity of hot-melt extrusion
Authors
Keywords
Hot-melt extrusion, Multicomponent systems, Co-crystals, Co-amorphous systems, Pharmaceutical salts, Physicochemical properties
Journal
JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY
Volume 61, Issue -, Pages 102209
Publisher
Elsevier BV
Online
2020-11-10
DOI
10.1016/j.jddst.2020.102209
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Continuous twin screw granulation – An advanced alternative granulation technology for use in the pharmaceutical industry
- (2020) Suresh Bandari et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Polymer-Assisted Aripiprazole–Adipic Acid Cocrystals Produced by Hot Melt Extrusion Techniques
- (2020) Arun Butreddy et al. CRYSTAL GROWTH & DESIGN
- Continuous Manufacturing of Ketoprofen Delayed Release Pellets Using Melt Extrusion Technology: Application of QbD Design Space, Inline Near Infrared, and Inline Pellet Size Analysis
- (2020) Anh Q. Vo et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Formulation Optimization for Gastroretentive Drug Delivery System of Carvedilol Cocrystals Using Design of Experiment
- (2019) Gasper J. Fernandes et al. Journal of Pharmaceutical Innovation
- Impact of polymeric excipient on cocrystal formation via hot-melt extrusion and subsequent downstream processing
- (2019) Maryam Karimi-Jafari et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Continuous, simultaneous cocrystallization and formulation of Theophylline and 4-Aminobenzoic acid pharmaceutical cocrystals using twin screw melt granulation
- (2019) Rahamatullah Shaikh et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Tuning the cocrystal yield in matrix-assisted cocrystallisation via hot melt extrusion: A case of theophylline-nicotinamide cocrystal
- (2019) Maciej Gajda et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Pharmaceutical cocrystals of naringenin with improved dissolution performance
- (2018) Chun Luo et al. CRYSTENGCOMM
- Optimising the in vitro and in vivo performance of oral cocrystal formulations via spray coating
- (2018) Dolores R. Serrano et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- The role of the polymer matrix in solvent-free hot melt extrusion continuous process for mechanochemical synthesis of pharmaceutical cocrystal
- (2018) Maciej Gajda et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Melt extrusion with poorly soluble drugs – An integrated review
- (2018) Michael A. Repka et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Hot Melt Extrusion: Highlighting Physicochemical Factors to Be Investigated While Designing and Optimizing a Hot Melt Extrusion Process
- (2018) Roberta Censi et al. Pharmaceutics
- Preparation of a crystalline salt of indomethacin and tromethamine by hot melt extrusion technology
- (2018) Mustafa Bookwala et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Engineering of pharmaceutical cocrystals in an excipient matrix: Spray drying versus hot melt extrusion
- (2018) David Walsh et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Coprocessing of Pharmaceutical Cocrystals for High Quality and Enhanced Physicochemical Stability
- (2018) Steven A. Ross et al. CRYSTAL GROWTH & DESIGN
- Mechanochemical Synthesis of Carvedilol Cocrystals Utilizing Hot Melt Extrusion Technology
- (2018) Gasper J. Fernandes et al. Journal of Pharmaceutical Innovation
- Hot Melt Extrusion and Spray Drying of Co-amorphous Indomethacin-Arginine With Polymers
- (2017) Elisabeth Lenz et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Mechanochemical Synthesis of Pharmaceutical Cocrystal Suspensions via Hot Melt Extrusion: Enhancing Cocrystal Yield
- (2017) Shu Li et al. MOLECULAR PHARMACEUTICS
- Continuous Preparation of 1:1 Haloperidol–Maleic Acid Salt by a Novel Solvent-Free Method Using a Twin Screw Melt Extruder
- (2017) Hung Lin Lee et al. MOLECULAR PHARMACEUTICS
- Melt Extrusion of High-Dose Co-Amorphous Drug-Drug Combinations
- (2017) Lærke Arnfast et al. PHARMACEUTICAL RESEARCH
- Pharmaceutical cocrystals: along the path to improved medicines
- (2016) Naga K. Duggirala et al. CHEMICAL COMMUNICATIONS
- Continuous Manufacturing of High Quality Pharmaceutical Cocrystals Integrated with Process Analytical Tools for In-Line Process Control
- (2016) Hiren G. Moradiya et al. CRYSTAL GROWTH & DESIGN
- Multidrug co-crystals: towards the development of effective therapeutic hybrids
- (2016) Rajesh Thipparaboina et al. DRUG DISCOVERY TODAY
- Rational excipient selection for co-amorphous formulations
- (2016) Ossi Korhonen et al. Expert Opinion on Drug Delivery
- Mechanochemical Synthesis of Pharmaceutical Cocrystal Suspensions via Hot Melt Extrusion: Feasibility Studies and Physicochemical Characterization
- (2016) Shu Li et al. MOLECULAR PHARMACEUTICS
- Identification of New Cocrystal Systems with Stoichiometric Diversity of Salicylic Acid Using Thermal Methods
- (2016) Zhengzheng Zhou et al. PHARMACEUTICAL RESEARCH
- Powder grinding preparation of co-amorphous β-azelnidipine and maleic acid combination: Molecular interactions and physicochemical properties
- (2016) Yazhu Han et al. POWDER TECHNOLOGY
- Disappearing Polymorphs Revisited
- (2015) Dejan-Krešimir Bučar et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- How Development and Manufacturing Will Need to Be Structured—Heads of Development/Manufacturing May 20–21, 2014 Continuous Manufacturing Symposium
- (2015) Kevin Nepveux et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Regulatory and Quality Considerations for Continuous Manufacturing May 20–21, 2014 Continuous Manufacturing Symposium
- (2015) Gretchen Allison et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Achieving Continuous Manufacturing for Final Dosage Formation: Challenges and How to Meet Them May 20–21 2014 Continuous Manufacturing Symposium
- (2015) Stephen Byrn et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- A Strategy for Co-former Selection to Design Stable Co-amorphous Formations Based on Physicochemical Properties of Non-steroidal Inflammatory Drugs
- (2015) Hiroshi Ueda et al. PHARMACEUTICAL RESEARCH
- Process Analytical Technology for continuous manufacturing of solid-dosage forms
- (2015) Margot Fonteyne et al. TRAC-TRENDS IN ANALYTICAL CHEMISTRY
- Continuous cocrystallisation of carbamazepine and trans-cinnamic acid via melt extrusion processing
- (2014) Hiren G. Moradiya et al. CRYSTENGCOMM
- Preparation and characterization of co-amorphous Ritonavir–Indomethacin systems by solvent evaporation technique: Improved dissolution behavior and physical stability without evidence of intermolecular interactions
- (2014) Swapnil J. Dengale et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Application of twin screw extrusion to the manufacture of cocrystals: scale-up of AMG 517–sorbic acid cocrystal production
- (2014) Dominick Daurio et al. FARADAY DISCUSSIONS
- Novel pharmaceutical cocrystal consisting of paracetamol and trimethylglycine, a new promising cocrystal former
- (2014) Yusuke Maeno et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Matrix-Assisted Cocrystallization (MAC) Simultaneous Production and Formulation of Pharmaceutical Cocrystals by Hot-Melt Extrusion
- (2014) Kevin Boksa et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Development of sustained-release formulations processed by hot-melt extrusion by using a quality-by-design approach
- (2014) Muhammad T. Islam et al. Drug Delivery and Translational Research
- Amino acids as co-amorphous stabilizers for poorly water soluble drugs – Part 1: Preparation, stability and dissolution enhancement
- (2013) Korbinian Löbmann et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Amino acids as co-amorphous stabilizers for poorly water-soluble drugs – Part 2: Molecular interactions
- (2013) Korbinian Löbmann et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Coamorphous repaglinide–saccharin with enhanced dissolution
- (2013) Yuan Gao et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Process monitoring and visualization solutions for hot-melt extrusion: a review
- (2013) Lien Saerens et al. JOURNAL OF PHARMACY AND PHARMACOLOGY
- Proliposomes of lisinopril dihydrate for transdermal delivery: Formulation aspects and evaluation
- (2013) Suresh Bandari et al. KOREAN JOURNAL OF CHEMICAL ENGINEERING
- Drug–Drug Coamorphous Systems: Characterization and Physicochemical Properties of Coamorphous Atorvastatin with Carvedilol and Glibenclamide
- (2013) Ali Shayanfar et al. Journal of Pharmaceutical Innovation
- Characterization of Non-stoichiometric Hydration and the Dehydration Behavior of Sitafloxacin Hydrate
- (2012) Tetsuya Suzuki et al. CHEMICAL & PHARMACEUTICAL BULLETIN
- Regime map development for continuous twin screw granulation
- (2012) Wei-Da Tu et al. CHEMICAL ENGINEERING SCIENCE
- Polymorphs, Salts, and Cocrystals: What’s in a Name?
- (2012) Srinivasulu Aitipamula et al. CRYSTAL GROWTH & DESIGN
- Acid–base crystalline complexes and the pKa rule
- (2012) Aurora J. Cruz-Cabeza CRYSTENGCOMM
- Twin screw wet granulation: The study of a continuous twin screw granulator using Positron Emission Particle Tracking (PEPT) technique
- (2012) Kai T. Lee et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Co-amorphous simvastatin and glipizide combinations show improved physical stability without evidence of intermolecular interactions
- (2012) Korbinian Löbmann et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Establishment of cocrystal cocktail grinding method for rational screening of pharmaceutical cocrystals
- (2012) Katsuhiko Yamamoto et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Thermal analysis and FTIR spectral curve-fitting investigation of formation mechanism and stability of indomethacin-saccharin cocrystals via solid-state grinding process
- (2012) Gang-Chun Zhang et al. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS
- Rational Coformer or Solvent Selection for Pharmaceutical Cocrystallization or Desolvation
- (2012) Yuriy A. Abramov et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Real-time and in situ monitoring of mechanochemical milling reactions
- (2012) Tomislav Friščić et al. Nature Chemistry
- Twin screw wet granulation: Influence of formulation parameters on granule properties and growth behavior
- (2012) A.S. El Hagrasy et al. POWDER TECHNOLOGY
- Twin screw granulation using conveying screws: Effects of viscosity of granulation liquids and flow of powders
- (2012) Ranjit M. Dhenge et al. POWDER TECHNOLOGY
- Single Particle Nonlinear Optical Imaging of Trace Crystallinity in an Organic Powder
- (2011) D. Wanapun et al. ANALYTICAL CHEMISTRY
- Hansen solubility parameter as a tool to predict cocrystal formation
- (2011) Mohammad Amin Mohammad et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Pharmaceutical cocrystals: An overview
- (2011) Ning Qiao et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Cocrystallization and amorphization induced by drug–excipient interaction improves the physical properties of acyclovir
- (2011) Takaaki Masuda et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Prediction of the Thermal Phase Diagram of Amorphous Solid Dispersions by Flory–Huggins Theory
- (2011) Yinyan Zhao et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Coamorphous Drug Systems: Enhanced Physical Stability and Dissolution Rate of Indomethacin and Naproxen
- (2011) Korbinian Löbmann et al. MOLECULAR PHARMACEUTICS
- Improving the Chemical Stability of Amorphous Solid Dispersion with Cocrystal Technique by Hot Melt Extrusion
- (2011) Xu Liu et al. PHARMACEUTICAL RESEARCH
- Virtual cocrystal screening
- (2011) Daniele Musumeci et al. Chemical Science
- Application of Twin Screw Extrusion in the Manufacture of Cocrystals, Part I: Four Case Studies
- (2011) Dominick Daurio et al. Pharmaceutics
- The Utility of Sulfonate Salts in Drug Development
- (2010) David P. Elder et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Physical Stability of Salts of Weak Bases in the Solid-State
- (2010) Gregory A. Stephenson et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Study of the Amorphous Glibenclamide Drug: Analysis of the Molecular Dynamics of Quenched and Cryomilled Material
- (2010) Z. Wojnarowska et al. MOLECULAR PHARMACEUTICS
- Enabling the Intestinal Absorption of Highly Polar Antiviral Agents: Ion-Pair Facilitated Membrane Permeation of Zanamivir Heptyl Ester and Guanidino Oseltamivir
- (2010) Jonathan M. Miller et al. MOLECULAR PHARMACEUTICS
- Cocrystalization and Simultaneous Agglomeration Using Hot Melt Extrusion
- (2010) Ravindra S. Dhumal et al. PHARMACEUTICAL RESEARCH
- Crystal Structure Transformations and Dissolution Studies of Cimetidine–Piroxicam Coprecipitates and Physical Mixtures
- (2009) Vimon Tantishaiyakul et al. AAPS PHARMSCITECH
- Cambridge Structural Database Analysis of Molecular Complementarity in Cocrystals
- (2009) László Fábián CRYSTAL GROWTH & DESIGN
- Quasi-equilibrium analysis of the ion-pair mediated membrane transport of low-permeability drugs
- (2009) Jonathan M. Miller et al. JOURNAL OF CONTROLLED RELEASE
- Enhanced dissolution rate and synchronized release of drugs in binary systems through formulation: Amorphous naproxen–cimetidine mixtures prepared by mechanical activation
- (2009) Morten Allesø et al. JOURNAL OF CONTROLLED RELEASE
- Manufacture of pharmaceutical co‐crystals using twin screw extrusion: A solvent‐less and scalable process
- (2009) Cesar Medina et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Wet Granulation in a Twin‐Screw Extruder: Implications of Screw Design
- (2009) M.R. Thompson et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- A rapid thermal method for cocrystal screening
- (2008) Enxian Lu et al. CRYSTENGCOMM
- Influence of particle size and preparation methods on the physical and chemical stability of amorphous simvastatin
- (2008) F ZHANG et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Physical characterization and stability of amorphous indomethacin and ranitidine hydrochloride binary systems prepared by mechanical activation
- (2008) N CHIENG et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Effect of Water Activity on the Transformation between Hydrate and Anhydrate of Carbamazepine
- (2008) Yi Li et al. ORGANIC PROCESS RESEARCH & DEVELOPMENT
Find the ideal target journal for your manuscript
Explore over 38,000 international journals covering a vast array of academic fields.
SearchCreate your own webinar
Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.
Create Now