Novel 3-Acetyl-2,5-disubstituted-1,3,4-oxadiazolines: Synthesis and Biological Activity

Synthesis and in Vitro Antimicrobial Activity Screening of New 3‐Acetyl‐2,5‐disubstituted‐1,3,4‐oxadiazoline Derivatives

(2019) Łukasz Popiołek et al.   CHEMISTRY & BIODIVERSITY

Synthesis, in vitro antibacterial and antifungal evaluation of novel 1,3,4-oxadiazole thioether derivatives bearing the 6-fluoroquinazolinylpiperidinyl moiety

(2019) Jun Shi et al.   CHINESE CHEMICAL LETTERS

Antimicrobial and antiprotozoal activity of 3-acetyl-2,5-disubstituted-1,3,4-oxadiazolines: a review

(2019) Kinga Paruch et al.   MEDICINAL CHEMISTRY RESEARCH

New hydrazide-hydrazones of isonicotinic acid: synthesis, lipophilicity and in vitro antimicrobial screening

(2018) Łukasz Popiołek et al.   Chemical Biology & Drug Design

Antimicrobial activity of 1,3,4-oxadiazole derivatives against planktonic cells and biofilm of Staphylococcus aureus

(2018) Zhaojun Zheng et al.   Future Medicinal Chemistry

Synthesis, characterization and pharmacological evaluation of (Z)-2-(5-(biphenyl-4-yl)-3-(1-(imino)ethyl)-2,3-dihydro-1,3,4-oxadiazol-2-yl)phenol derivatives as potent antimicrobial and antioxidant agents

(2017) Manav Malhotra et al.   Arabian Journal of Chemistry

Synthesis and molecular modeling studies of novel pyrrole analogs as antimycobacterial agents

(2017) Shrinivas D. Joshi et al.   Journal of Saudi Chemical Society

Methicillin-Resistant Staphylococcus epidermidis Is Part of the Skin Flora on the Hands of Both Healthy Individuals and Hospital Workers

(2016) Kiyoshi Watanabe et al.   BIOLOGICAL & PHARMACEUTICAL BULLETIN

Design, synthesis, andin vitroantimicrobial activity of hydrazide-hydrazones of 2-substituted acetic acid

(2016) Łukasz Popiołek et al.   Chemical Biology & Drug Design

Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold

(2016) Simona Distinto et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2,5-Disubstituted 1,3,4-oxadiazole derivatives of chromeno[4,3-b]pyridine: synthesis and study of antimicrobial potency

(2016) Ghanshyam R. Jadhav et al.   HETEROCYCLIC COMMUNICATIONS

Conventional and microwave techniques for the synthesis and antimicrobial studies of novel 1-[2-(2-chloro-6-methyl(3-quinolyl))-5-(4-nitrophenyl)-(1,3,4-oxadiazolin-3-yl)]-3-(aryl)prop-2-en-1-ones

(2016) N.C. Desai et al.   Arabian Journal of Chemistry

N-(1′-naphthyl)-3,4,5-trimethoxybenzohydrazide as microtubule destabilizer: Synthesis, cytotoxicity, inhibition of cell migration and in vivo activity against acute lymphoblastic leukemia

(2015) Lívia B. Salum et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Exploring 5-nitrofuran derivatives against nosocomial pathogens: Synthesis, antimicrobial activity and chemometric analysis

(2014) Rodrigo Rocha Zorzi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological evaluation of new oxadiazoline-substituted naphthalenyl acetates as anticancer agents

(2014) Ibrahim Chaaban et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Discovery and Characterization of Potent Thiazoles versus Methicillin- and Vancomycin-Resistant Staphylococcus aureus

(2014) Haroon Mohammad et al.   JOURNAL OF MEDICINAL CHEMISTRY

5-Nitro-2-furfuriliden derivatives as potential anti-Trypanosoma cruzi agents: Design, synthesis, bioactivity evaluation, cytotoxicity and exploratory data analysis

(2013) Fanny Palace-Berl et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, characterization and molecular docking studies of some new 1,3,4-oxadiazolines bearing 6-methylpyridine moiety for antimicrobial property

(2013) P.C. Shyma et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Phase III, Randomized, Placebo-Controlled Study of Docetaxel in Combination With Zibotentan in Patients With Metastatic Castration-Resistant Prostate Cancer

(2013) Karim Fizazi et al.   JOURNAL OF CLINICAL ONCOLOGY

Nitrogen heterocycles as potential monoamine oxidase inhibitors: Synthetic aspects

(2013) Pravin O. Patil et al.   Arabian Journal of Chemistry

Synthesis, molecular modeling and preliminary biological evaluation of a set of 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazole as potential antibacterial, anti-Trypanosoma cruzi and antifungal agents

(2011) Marina Ishii et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, spectroscopy and electrochemistry of new 4-(4-acetyl-5- substituted-4, 5-dihydro-1, 3,4-oxodiazol-2-yl)methoxy)-2H-chromen-2-ones as a novel class of potential antibacterial and antioxidant derivatives

(2011) N. Hamdi et al.   COMPTES RENDUS CHIMIE

3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A New Scaffold for the Selective Inhibition of Monoamine Oxidase B

(2011) Elias Maccioni et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Bioactivity of Novel Bis-heterocyclic Compounds Containing Pyrazole and Oxadiazoline

(2011) Jin-Feng Yang et al.   JOURNAL OF THE CHINESE CHEMICAL SOCIETY

Synthesis and biological activity of hydrazide–hydrazones and their corresponding 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazoles

(2011) Bedia Koçyiğit-Kaymakçıoğlu et al.   MEDICINAL CHEMISTRY RESEARCH

Synthesis of some novel 2-substituted-5-[isopropylthiazole] clubbed 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents

(2010) G.V. Suresh Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Microwave-assisted efficient synthesis of glucose-based 3-acetyl-5-alkyl-2,3-dihydro-1,3,4-oxadiazole derivatives catalyzed by sodium acetate

(2009) Lin-Na Wang et al.   CARBOHYDRATE RESEARCH

Synthesis and Antimicrobial Evaluation of Some New Oxadiazoles Derived from Phenylpropionohydrazides

(2009) Neeraj Kumar Fuloria et al.   MOLECULES

1,3,4-Oxadiazole-3(2H)-carboxamide derivatives as potential novel class of monoamine oxidase (MAO) inhibitors: Synthesis, evaluation, and role of urea moiety

(2008) Shaoyong Ke et al.   BIOORGANIC & MEDICINAL CHEMISTRY

1,3,4-Oxadiazoline derivatives as novel potential inhibitors targeting chitin biosynthesis: Design, synthesis and biological evaluation

(2008) Shaoyong Ke et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Raltegravir: The first HIV integrase inhibitor

(2008) Jennifer Cocohoba et al.   CLINICAL THERAPEUTICS

Synthesis of new 4-pyrrol-1-yl benzoic acid hydrazide analogs and some derived oxadiazole, triazole and pyrrole ring systems: A novel class of potential antibacterial and antitubercular agents

(2007) S.D. Joshi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY