A straightforward access to 3-trifluoromethyl-1H-indazoles via (3+2)-cycloaddition of arynes with nitrile imines derived from trifluoroacetonitrile

The Huisgen Reaction: Milestones of the 1,3‐Dipolar Cycloaddition

(2020) Martin Breugst et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly fluorinated 2,3-dihydro-1,3,4-thiadiazole derivatives via [3+2]-cycloadditions of tertiary thioamides with nitrile imines derived from trifluoroacetonitrile

(2020) Greta Utecht-Jarzyńska et al.   JOURNAL OF FLUORINE CHEMISTRY

Trapping of trifluoroacetonitrile imines with mercaptoacetaldehyde and mercaptocarboxylic acids: An access to fluorinated 1,3,4-thiadiazine derivatives via (3+3)-annulation

(2019) Greta Utecht-Jarzyńska et al.   JOURNAL OF FLUORINE CHEMISTRY

Synthesis of Pyrrolo[2,3-c]isoquinolines via the Cycloaddition of Benzyne with Arylideneaminopyrroles: Photophysical and Crystallographic Study

(2019) Juan-Carlos Castillo et al.   ACS Omega

Polysubstituted 3-trifluoromethylpyrazoles: regioselective (3 + 2)-cycloaddition of trifluoroacetonitrile imines with enol ethers and functional group transformations

(2018) Greta Utecht et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A Straightforward Access to Trifluoromethylated Spirobipyrazolines through a Double (3+2)-Cycloaddition of Fluorinated Nitrile Imines with Alkoxyallenes

(2018) Marcin Jasiński et al.   SYNLETT

Synthesis and evaluation of steroidal thiazoline conjugates as potential antiviral agents

(2018) Shaoyong Ke et al.   Future Medicinal Chemistry

Recent Advances in Indazole-Containing Derivatives: Synthesis and Biological Perspectives

(2018) Shu-Guang Zhang et al.   MOLECULES

Expected and unexpected results in reactions of fluorinated nitrile imines with (cyclo)aliphatic thioketones

(2017) Greta Utecht et al.   JOURNAL OF FLUORINE CHEMISTRY

First (3+2)-Cycloadditions of Thiochalcones as C=S Dipolarophiles: Efficient Synthesis of 1,3,4-Thiadiazoles via Reactions with Fluorinated Nitrile Imines

(2017) Grzegorz Mlostoń et al.   SYNTHESIS-STUTTGART

Fluorine-containing indazoles: Synthesis and biological activity

(2016) Galina N. Lipunova et al.   JOURNAL OF FLUORINE CHEMISTRY

Trifluoromethylated 2,3-dihydro-1,3,4-thiadiazoles via the regioselective [3+2]-cycloadditions of fluorinated nitrile imines with aryl, hetaryl, and ferrocenyl thioketones

(2016) Grzegorz Mlostoń et al.   JOURNAL OF FLUORINE CHEMISTRY

Inhibition of Mitochondrial Complex II by the Anticancer Agent Lonidamine

(2015) Lili Guo et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Tautomeric equilibrium in trifluoroacetaldehyde arylhydrazones

(2015) Agata Wojciechowska et al.   TETRAHEDRON

Aryne Cycloaddition Reactions in the Synthesis of Large Polycyclic Aromatic Compounds

(2013) Dolores Pérez et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Comprehensive History of Arynes in Natural Product Total Synthesis

(2012) Pamela M. Tadross et al.   CHEMICAL REVIEWS

New Synthesis of 1-Substituted-1H-indazoles via 1,3-Dipolar Cycloaddition ofin situGenerated Nitrile Imines and Benzyne

(2010) Christian Spiteri et al.   ORGANIC LETTERS

Fluorinated indazoles as novel selective inhibitors of nitric oxide synthase (NOS): Synthesis and biological evaluation

(2009) Rosa M. Claramunt et al.   BIOORGANIC & MEDICINAL CHEMISTRY

RECENT APPLICATIONS OF ARYNE CHEMISTRY TO ORGANIC SYNTHESIS. A REVIEW

(2009) Roberto Sanz   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

Gamendazole, an Orally Active Indazole Carboxylic Acid Male Contraceptive Agent, Targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and Stimulates Il1a Transcription in Rat Sertoli Cells1

(2008) Joseph S. Tash et al.   BIOLOGY OF REPRODUCTION