New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

1,2,3-Triazole-containing hybrids as leads in medicinal chemistry: A recent overview

(2019) Khurshed Bozorov et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Sulfamates in drug design and discovery: Pre-clinical and clinical investigations

(2019) Seyed-Omar Zaraei et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

New potent STS inhibitors based on fluorinated 4-(1-phenyl-1H-[1,2,3]triazol-4-yl)-phenyl sulfamates

(2019) Mateusz Daśko et al.   JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH

Boronic acid inhibitors of the class A β-lactamase KPC-2

(2018) Jingyuan Zhou et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Radiosynthesis and biological evaluation of 18 F-labeled 4-anilinoquinazoline derivative ( 18 F-FEA-Erlotinib) as a potential EGFR PET agent

(2018) Shun Huang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Hetero-Diels-Alder reactions of novel 3-triazolyl-nitrosoalkenes as an approach to functionalized 1,2,3-triazoles with antibacterial profile

(2018) Susana M.M. Lopes et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

18F-Positron Emitting/Trimethine Cyanine-Fluorescent Contrast for Image-Guided Prostate Cancer Management

(2018) Harikrishna Kommidi et al.   JOURNAL OF MEDICINAL CHEMISTRY

SULFATION PATHWAYS: Steroid sulphatase inhibition via aryl sulphamates: clinical progress, mechanism and future prospects

(2018) Barry V L Potter   JOURNAL OF MOLECULAR ENDOCRINOLOGY

Synthesis and Antimalarial Evaluation of [1, 2,3]-Triazole-Tethered Sulfonamide-Berberine Hybrids

(2018) Neha Batra et al.   ChemistrySelect

Sulfatase inhibitors for recidivist breast cancer treatment: A chemical review

(2016) Ramanpreet Shah et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent Developments of Steroid Sulfatase Inhibitors as Anti-Cancer Agents

(2012) Paul Foster et al.   Anti-Cancer Agents in Medicinal Chemistry

Irosustat: a first-generation steroid sulfatase inhibitor in breast cancer

(2011) Carlo Palmieri et al.   Expert Review of Anticancer Therapy

Steroid sulfatase: A pivotal player in estrogen synthesis and metabolism

(2011) Atul Purohit et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Increased estrogen sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1(17β-HSD1) following neoadjuvant aromatase inhibitor therapy in breast cancer patients

(2010) Niramol Chanplakorn et al.   BREAST CANCER RESEARCH AND TREATMENT

A New Therapeutic Strategy against Hormone-Dependent Breast Cancer: The Preclinical Development of a Dual Aromatase and Sulfatase Inhibitor

(2008) P. A. Foster et al.   CLINICAL CANCER RESEARCH