Bestatin and bacitracin inhibit porcine kidney cortex dipeptidyl peptidase IV activity and reduce human melanoma MeWo cell viability

Anti-diabetic drugs recent approaches and advancements

(2020) Jayanta Dowarah et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Dipeptidyl peptidase 4 inhibitors and their potential immune modulatory functions

(2020) Shiying Shao et al.   PHARMACOLOGY & THERAPEUTICS

Structure–activity relationships study on biological activity of peptides as dipeptidyl peptidase IV inhibitors by chemometric modeling

(2019) Paulina Kęska et al.   Chemical Biology & Drug Design

Bacitracin is a non-competitive inhibitor of porcine M1 family neutral and glutamyl aminopeptidases

(2019) Yarini Arrebola et al.   NATURAL PRODUCT RESEARCH

The role of renal dipeptidyl peptidase-4 in kidney disease: renal effects of dipeptidyl peptidase-4 inhibitors with a focus on linagliptin

(2018) Keizo Kanasaki   CLINICAL SCIENCE

Design of Aminopeptidase N Inhibitors as Anti-cancer Agents

(2018) Sk. Abdul Amin et al.   JOURNAL OF MEDICINAL CHEMISTRY

Critical role of Dipeptidyl Peptidase IV: A therapeutic target for cancer & diabetes

(2018) Priyankar Paira et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Role of ubenimex as an anticancer drug and its synergistic effect with Akt inhibitor in human A375 and A2058 cells

(2018) Xiaoqing Wang et al.   OncoTargets and Therapy

In Silico Approaches Applied to the Study of Peptide Analogs of Ile-Pro-Ile in Relation to Their Dipeptidyl Peptidase IV Inhibitory Properties

(2018) Alice B. Nongonierma et al.   Frontiers in Endocrinology

The MEROPS database of proteolytic enzymes, their substrates and inhibitors in 2017 and a comparison with peptidases in the PANTHER database

(2017) Neil D Rawlings et al.   NUCLEIC ACIDS RESEARCH

Recent approaches to medicinal chemistry and therapeutic potential of dipeptidyl peptidase-4 (DPP-4) inhibitors

(2014) Bhumika D. Patel et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A comparative study of the binding modes of recently launched dipeptidyl peptidase IV inhibitors in the active site

(2013) Mika Nabeno et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Protein disulfide isomerase: a promising target for cancer therapy

(2013) Shili Xu et al.   DRUG DISCOVERY TODAY

Effect of zinc and calcium ions on the rat kidney membrane-bound form of dipeptidyl peptidase IV

(2013) Hansel Gómez et al.   JOURNAL OF BIOSCIENCES

Dipeptidyl peptidase-4 inhibitors: Multitarget drugs, not only antidiabetes drugs (D ipeptidyl peptidase -4抑制剂：多靶点药物，不仅仅是降糖药)

(2013) Yunjuan Zhao et al.   Journal of Diabetes

Identification of diverse dipeptidyl peptidase IV inhibitors via structure-based virtual screening

(2012) Cui Li et al.   JOURNAL OF MOLECULAR MODELING

Dipeptidyl peptidase IV, aminopeptidase N and DPIV/APN-like proteases in cerebral ischemia

(2012) Peter Röhnert et al.   Journal of Neuroinflammation

Avogadro: an advanced semantic chemical editor, visualization, and analysis platform

(2012) Marcus D Hanwell et al.   Journal of Cheminformatics

Synthesis of New (−)-Bestatin-Based Inhibitor Libraries Reveals a Novel Binding Mode in the S1 Pocket of the Essential Malaria M1 Metalloaminopeptidase

(2011) Geetha Velmourougane et al.   JOURNAL OF MEDICINAL CHEMISTRY

Bestatin-based chemical biology strategy reveals distinct roles for malaria M1- and M17-family aminopeptidases

(2011) M. B. Harbut et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Metallo-aminopeptidase inhibitors

(2010) Artur Mucha et al.   BIOCHIMIE

Aminopeptidase N (CD13) as a target for cancer chemotherapy

(2010) Malin Wickström et al.   CANCER SCIENCE

A Time-Resolved Fluorescence Probe for Dipeptidyl Peptidase 4 and Its Application in Inhibitor Screening

(2010) Mitsuyasu Kawaguchi et al.   CHEMISTRY-A EUROPEAN JOURNAL

The dipeptidyl peptidase IV family in cancer and cell biology

(2010) Denise M. T. Yu et al.   FEBS Journal

Recent insights into the role of dipeptidyl aminopeptidase IV (DPIV) and aminopeptidase N (APN) families in immune functions

(2009) Siegfried Ansorge et al.   CLINICAL CHEMISTRY AND LABORATORY MEDICINE

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

(2009) Garrett M. Morris et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY

Development of bestatin-based activity-based probes for metallo-aminopeptidases

(2008) Michael B. Harbut et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Increasing Melanoma Cell Death Using Inhibitors of Protein Disulfide Isomerases to Abrogate Survival Responses to Endoplasmic Reticulum Stress

(2008) P. E. Lovat et al.   CANCER RESEARCH

The ectopeptidases dipeptidyl peptidase IV (DP IV) and aminopeptidase N (APN) and their related enzymes as possible targets in the treatment of skin diseases

(2007) Anja Thielitz   Frontiers in Bioscience-Landmark

DP IV/CD26, APN/CD13 and related enzymes as regulators of T cell immunity: implications for experimental encephalomyelitis and multiple sclerosis

(2007) Dirk Reinhold   Frontiers in Bioscience-Landmark