Updating the CSIC Reaction (2003–2020)

An unexpected synthesis of β-amino-α-mesyl-γ-sultams upon mesylation of hindered α-aminonitriles

(2020) Maksim S. Dyachenko et al.   Chemistry of Heterocyclic Compounds

Synthesis of 4,4‐Disubstituted 1,2‐Thiazinane‐5‐one 1,1‐Dioxides via the CSIC [≠] Reaction Strategy

(2020) Maksim S. Dyachenko et al.   ChemistrySelect

Development of oxathiino[6,5-b]pyridine 2,2-dioxide derivatives as selective inhibitors of tumor-related carbonic anhydrases IX and XII

(2020) Aiga Grandāne et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthetic Approach to Fused Azasultams with 1,2,4-Thiadiazepine Framework

(2020) Demyd S. Milokhov et al.   SYNTHESIS-STUTTGART

Expected and unforeseen reactions of 2,3,3-trimethyl-1λ6-isothiazolidine-1,1,4-trione and their spiro derivative

(2019) Maria V. Popova et al.   TETRAHEDRON

Synthesis, X-ray crystal and monoamine oxidase inhibitory activity of 4,6-dihydrobenzo[c]pyrano[2,3-e][1,2]thiazine 5,5-dioxides: In vitro studies and docking analysis

(2019) Shakeel Ahmad et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

Synthesis of Novel 3  a ‐Substituted Tetrahydro‐1 H ‐1λ 6 ‐pyrrolo[1,2‐ b ]isothiazole‐1,1,3(2 H )‐triones through the CSIC Reaction

(2019) Taras V. Omelian et al.   ChemistrySelect

Synthesis, characterization, monoamine oxidase inhibition, molecular docking and dynamic simulations of novel 2,1-benzothiazine-2,2-dioxide derivatives

(2018) Shakeel Ahmad et al.   BIOORGANIC CHEMISTRY

Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies

(2018) Alessio Nocentini et al.   CHEMISTRY-A EUROPEAN JOURNAL

4-Amino-2,3-dihydro-1λ6-isothiazole-1,1-dioxides and their chemical properties evaluation

(2018) Maksim S. Dyachenko et al.   MOLECULAR DIVERSITY

The simplest synthesis of 5,5-disubstituted and spiranic methyl 4-amino-2,2-dioxo-2,5-dihydro-1,2λ 6 -oxathiole-3-carboxylates

(2018) Alexey V. Dobrydnev et al.   TETRAHEDRON LETTERS

One-pot synthesis of methyl 4-amino-2,3,3-trisubstituted-1,1-dioxo-2,3-dihydro-1H-1λ6-isothiazole-5-carboxylates

(2018) Alexey V. Dobrydnev et al.   MONATSHEFTE FUR CHEMIE

Synthesis of phosphorus analogs of TSAO-T

(2018) Marina Moura et al.   TETRAHEDRON

Progress in the synthesis of δ-sultones

(2017) Christina Gaunersdorfer et al.   MONATSHEFTE FUR CHEMIE

Synthesis of a series of tetraminic acid sulfone analogs

(2017) Maria V. Popova et al.   MONATSHEFTE FUR CHEMIE

Iridium-Catalyzed Asymmetric Hydrogenation of 2H-Chromenes: A Highly Enantioselective Approach to Isoflavan Derivatives

(2017) Jingzhao Xia et al.   ORGANIC LETTERS

Catalytic Asymmetric Direct-Type 1,4-Addition Reactions of Alkanesulfonamides

(2017) Shū Kobayashi et al.   SYNLETT

Structure and function of carbonic anhydrases

(2016) C. T. Supuran   BIOCHEMICAL JOURNAL

Reactivity, Selectivity, and Stability in Sulfenic Acid Detection: A Comparative Study of Nucleophilic and Electrophilic Probes

(2016) Vinayak Gupta et al.   BIOCONJUGATE CHEMISTRY

Discovery of (2-benzoylethen-1-ol)-containing 1,2-benzothiazine derivatives as novel 4-hydroxyphenylpyruvate dioxygenase (HPPD) inhibiting-based herbicide lead compounds

(2016) Kang Lei et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Profiling the reactivity of cyclic C-nucleophiles towards electrophilic sulfur in cysteine sulfenic acid

(2016) Vinayak Gupta et al.   Chemical Science

Peculiarities of 2-amino-3-R-4-aryl-4H-pyranes multicomponent synthesis derived from 1H-2,1-benzothiazin-4(3H)-one 2,2-dioxide

(2016) Dmitry A. Lega et al.   RSC Advances

Sultones and Sultines via a Julia-Kocienski Reaction of Epoxides

(2015) Geoffrey M. T. Smith et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free Allene-Based Synthesis of Enantiopure Fused Polycyclic Sultones

(2015) Benito Alcaide et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of the First Representatives of Spiro-1λ6-isothiazolidine-1,1,4-triones

(2015) Alexey Dobrydnev et al.   SYNTHESIS-STUTTGART

Synthesis and anti-BVDV activity of novel δ-sultones in vitro: Implications for HCV therapies

(2014) Hai-Wei Xu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

2,1-Benzothiazine 2,2-Dioxides. 5*. Hydrolysis of Alkyl 1-R-4-Hydroxy-2,2-Dioxo-1Н-2λ6,1-Benzo-Thiazine-3-Carboxylates**

(2014) I. V. Ukrainets et al.   Chemistry of Heterocyclic Compounds

2,1-Benzothiazine 2,2-Dioxides. 8*. Synthesis and Structure of 2'-Amino-2-Oxo-1,2-Dihydro-6'H-Spiro-[Indole-3,4'-Pyrano[3,2-c][2,1]Benzothiazine]-3'-Carbonitrile 5',5'-Dioxides

(2014) I. V. Ukrainets et al.   Chemistry of Heterocyclic Compounds

Synthesis of 5-Amino-3,3-dimethyl-7-phenyl-3H-[1,2]oxathiolo[4,3-b]pyridine-6-carbonitrile 1,1-Dioxides

(2014) Mourad Chioua et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

An efficient, three-component synthesis and molecular structure of derivatives of 2-amino-3-R-6-ethyl-4,6-dihydropyrano[3,2-c][2,1]benzothiazine-5,5-dioxide spirocombined with a 2-oxindole nucleus

(2014) Leonid A. Shemchuk et al.   TETRAHEDRON

Structure-based discovery of cellular-active allosteric inhibitors of FAK

(2013) Naoki Tomita et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

2,1-Benzothiazine 2,2-Dioxides. 1. Synthesis, Structure, and Analgesic Activity of 1-R-4-Hydroxy-2,2-Dioxo-1H-2λ6,1-Benzothiazine-3-Carboxylic Acid Esters

(2013) I. V. Ukrainets et al.   Chemistry of Heterocyclic Compounds

Regioselective Sulfonylation and N- to O-Sulfonyl Migration of Quinazolin-4(3H)-ones and Analogous Thienopyrimidin-4(3H)-ones

(2013) Matthias D. Mertens et al.   JOURNAL OF ORGANIC CHEMISTRY

Preparation of Spiro[4.4]oxaphospholene and -azaphospholene Systems from Carbohydrate Templates

(2013) Marina Moura et al.   JOURNAL OF ORGANIC CHEMISTRY

A new synthesis of sultams from amino alcohols

(2013) Nitin Lad et al.   TETRAHEDRON LETTERS

Recent Developments in the Synthesis and Application of Sultones

(2012) Shovan Mondal   CHEMICAL REVIEWS

Discovery and characterization of novel allosteric FAK inhibitors

(2012) Misa Iwatani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Access to a Wide Range of Sultams by Cyclodialkylation of α-Substituted Methanesulfonanilides

(2012) Valentin A. Rassadin et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Facile synthesis of coumarin bioisosteres—1,2-benzoxathiine 2,2-dioxides

(2012) Aiga Grandane et al.   TETRAHEDRON

From β-Amino-γ-sultone to Unusual Bicyclic Pyridine and Pyrazine Heterocyclic Systems: Synthesis and Cytostatic and Antiviral Activities

(2011) Sonia de Castro et al.   ChemMedChem

Lead Generation and Optimization Based on Protein-Ligand Complementarity

(2010) Koji Ogata et al.   MOLECULES

Dimethylformamide dimethyl acetal as a building block in heterocyclic synthesis

(2009) Fathi A. Abu-Shanab et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

4-Benzyloxy-γ-Sultone Derivatives: Discovery of a Novel Family of Non-Nucleoside Inhibitors of Human Cytomegalovirus and Varicella Zoster Virus

(2009) Sonia De Castro et al.   JOURNAL OF MEDICINAL CHEMISTRY

4-Benzyloxy-γ-Sultone Derivatives: Discovery of a Novel Family of Non-Nucleoside Inhibitors of Human Cytomegalovirus and Varicella Zoster Virus

(2009) Sonia De Castro et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and anti-HIV1 biological activity of novel 5″-ATSAO compounds

(2008) Cyrille Tomassi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Tetramic and tetronic acids: An update on new derivatives and biological aspects

(2008) Rainer Schobert et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Reactivity of the 4-Amino-5H-1,2-Oxathiole-2,2-Dioxide Heterocyclic System: A Combined Experimental and Theoretical Study

(2008) Sonia de Castro et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Useful Pd-Catalyzed Negishi Coupling Approach to Benzylic Sulfonamide Derivatives

(2008) Gang Zhou et al.   ORGANIC LETTERS

Halovinyl aldehydes: useful tools in organic synthesis

(2008) Sulagna Brahma et al.   TETRAHEDRON

A solid-phase synthetic method for 3,4-dihydro-1H-2,1-benzothiazin-4-one 2,2-dioxide derivatives

(2008) Moon-Kook Jeon et al.   TETRAHEDRON