Design, Synthesis, In Vitro and In Silico Studies of New Thiazolylhydrazine-Piperazine Derivatives as Selective MAO-A Inhibitors

“Design, Synthesis, Mechanistic Studies and In Silico ADME predictions of Benzimidazole derivatives as Novel Antifungal Agents”

(2020) Martha M. Morcoss et al.   BIOORGANIC CHEMISTRY

Discovery, synthesis, biological evaluation and molecular docking study of (R)-5-methylmellein and its analogs as selective monoamine oxidase A inhibitors

(2019) Chao Huang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of novel 2,3-dihydro-1H-inden-1-amine derivatives as selective monoamine oxidase B inhibitors

(2019) Shiyu Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

1,3,4-Oxadiazol-2-ylbenzenesulfonamides as privileged structures for the inhibition of monoamine oxidase B

(2019) Anton Shetnev et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design, synthesis and biological assessment of new thiazolylhydrazine derivatives as selective and reversible h MAO-A inhibitors

(2018) Nafiz Öncü Can et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

In vitro and in silico evaluation of new thiazole compounds as monoamine oxidase inhibitors

(2018) Begüm Nurpelin Sağlık et al.   BIOORGANIC CHEMISTRY

MAO enzymes inhibitory activity of new benzimidazole derivatives including hydrazone and propargyl side chains

(2017) Özgür Devrim Can et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Biological Evaluation of New Thiosemicarbazone Derivative Schiff Bases as Monoamine Oxidase Inhibitory Agents

(2017) Betül Çavuşoğlu et al.   MOLECULES

Synthesis of New Hydrazone Derivatives for MAO Enzymes Inhibitory Activity

(2017) Nafiz Öncü Can et al.   MOLECULES

Design and Synthesis of New Benzothiazole Compounds as Selective hMAO-B Inhibitors

(2017) Sinem Ilgın et al.   MOLECULES

SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules

(2017) Antoine Daina et al.   Scientific Reports

Design, synthesis, and AChE inhibitory activity of new benzothiazole–piperazines

(2016) Ümide Demir Özkay et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

( E )-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors

(2016) Nicoletta Desideri et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design and synthesis of novel chalcones as potent selective monoamine oxidase-B inhibitors

(2016) Arwa Hammuda et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of new donepezil analogues and investigation of their effects on cholinesterase enzymes

(2016) Begüm Nurpelin Sağlık et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines

(2012) Daniela Secci et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

admetSAR: A Comprehensive Source and Free Tool for Assessment of Chemical ADMET Properties

(2012) Feixiong Cheng et al.   Journal of Chemical Information and Modeling

Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors

(2010) Franco Chimenti et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors

(2010) Franco Chimenti et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Structure of human monoamine oxidase A at 2.2-A resolution: The control of opening the entry for substrates/inhibitors

(2008) S.-Y. Son et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA