Oral Administration of Peptide-Based Drugs: Beyond Lipinski's Rule

Rule of five in 2015 and beyond: Target and ligand structural limitations, ligand chemistry structure and drug discovery project decisions

(2016) Christopher A. Lipinski   ADVANCED DRUG DELIVERY REVIEWS

Quantifying the chameleonic properties of macrocycles and other high-molecular-weight drugs

(2016) Adrian Whitty et al.   DRUG DISCOVERY TODAY

Cell-Permeable Cyclic Peptides from Synthetic Libraries Inspired by Natural Products

(2015) William M. Hewitt et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oral Druggable Space beyond the Rule of 5: Insights from Drugs and Clinical Candidates

(2014) Bradley Croy Doak et al.   CHEMISTRY & BIOLOGY

The Emergence of Cyclic Peptides: The Potential of Bioengineered Peptide Drugs

(2014) Parashar Thapa et al.   International Journal of Peptide Research and Therapeutics

Physicochemical Descriptors of Aromatic Character and Their Use in Drug Discovery

(2014) Timothy J. Ritchie et al.   JOURNAL OF MEDICINAL CHEMISTRY

Form and Function in Cyclic Peptide Natural Products: A Pharmacokinetic Perspective

(2013) Andrew T. Bockus et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Macrocyclic Drugs and Clinical Candidates: What Can Medicinal Chemists Learn from Their Properties?

(2013) Fabrizio Giordanetto et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cyclic Peptides as Therapeutic Agents and Biochemical Tools

(2012) Sang-Hoon Joo   Biomolecules & Therapeutics

Therapeutic peptides

(2012) Fernando Albericio et al.   Future Medicinal Chemistry