α-Amylase Modulation: Discovery of Inhibitors Using a Multi-Pharmacophore Approach for Virtual Screening

Anthocyanin composition, antioxidant efficiency, and α-amylase inhibitor activity of different Hungarian sour cherry varieties (Prunus cerasus L.)

(2016) Judit R. Homoki et al.   FOOD CHEMISTRY

From carbohydrates to drug-like fragments: Rational development of novel α-amylase inhibitors

(2015) Jamil Al-Asri et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Inhibitory potency of flavonoid derivatives on influenza virus neuraminidase

(2014) Christin Rakers et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design, synthesis and molecular docking study of novel quinoxalin-2(1H)-ones as anti-tumor active agents with inhibition of tyrosine kinase receptor and studying their cyclooxygenase-2 activity

(2014) Shadia A. Galal et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Discovery of Sanggenon G as a natural cell-permeable small-molecular weight inhibitor of X-linked inhibitor of apoptosis protein (XIAP)

(2014) Maximilian A. Seiter et al.   FEBS Open Bio

Synthesis, biological activity and structure–activity relationships of new benzoic acid-based protein tyrosine phosphatase inhibitors endowed with insulinomimetic effects in mouse C2C12 skeletal muscle cells

(2013) Rosaria Ottanà et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Molecular Basis for the Recognition of Long-chain Substrates by Plant α-Glucosidases

(2013) Takayoshi Tagami et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Synthesis and glycosidase inhibitory activity of novel (2-phenyl-4H-benzopyrimedo[2,1-b]-thiazol-4-yliden)acetonitrile derivatives

(2012) Vijay S. Patil et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Computational Tools for In Silico Fragment-Based Drug Design

(2012) Jeremie Mortier et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Isolation of a New Phlorotannin, a Potent Inhibitor of Carbohydrate-Hydrolyzing Enzymes, from the Brown Alga Sargassum patens

(2012) Yasuko Kawamura-Konishi et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Order and Disorder: Differential Structural Impacts of Myricetin and Ethyl Caffeate on Human Amylase, an Antidiabetic Target

(2012) Leslie K. Williams et al.   JOURNAL OF MEDICINAL CHEMISTRY

Evaluation of Different Teas against Starch Digestibility by Mammalian Glycosidases

(2010) Lee Wah Koh et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Structures of human pancreatic α-amylase in complex with acarviostatins: Implications for drug design against type II diabetes

(2010) Xiaohong Qin et al.   JOURNAL OF STRUCTURAL BIOLOGY

The epidemic of type 2 diabetes mellitus in the Asia-Pacific region

(2010) Louis CK Low   PEDIATRIC DIABETES

Directed “in Situ” Inhibitor Elongation as a Strategy To Structurally Characterize the Covalent Glycosyl-Enzyme Intermediate of Human Pancreatic α-Amylase,

(2009) Ran Zhang et al.   BIOCHEMISTRY

How To Optimize Shape-Based Virtual Screening: Choosing the Right Query and Including Chemical Information

(2009) Johannes Kirchmair et al.   Journal of Chemical Information and Modeling

Evidence for pentagalloyl glucose binding to human salivary α-amylase through aromatic amino acid residues

(2008) Gyöngyi Gyémánt et al.   BIOCHIMICA ET BIOPHYSICA ACTA-PROTEINS AND PROTEOMICS

The Search for Novel Human Pancreatic α-Amylase Inhibitors: High-Throughput Screening of Terrestrial and Marine Natural Product Extracts

(2008) Chris A. Tarling et al.   CHEMBIOCHEM