16-Membered Macrolide Lactone Derivatives Bearing a Triazole-Functionalized Arm at the Aglycone C13 Position as Antibacterial and Anticancer Agents

Conversion of leucomycin-A3 antibiotic into novel triazole analogues via regio- and diastereoselective SN1′ substitution with allylic rearrangement and 1,3-dipolar cycloaddition of CuAAC type

(2016) Joanna Domagalska et al.   TETRAHEDRON LETTERS

Synthesis and antibacterial activity of a series of novel 9-O-acetyl- 4′-substituted 16-membered macrolides derived from josamycin

(2013) Zhehui Zhao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Transformation of josamycin in alkaline solution—intramolecular SN2 substitution or E1cB elimination and intramolecular Michael addition?

(2011) Piotr Przybylski et al.   TETRAHEDRON LETTERS

Preparation and biological evaluation of novel leucomycin analogs derived from nitroso Diels–Alder reactions

(2009) Baiyuan Yang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Unexpected α,β-unsaturated products of reductive amination of the macrolide antibiotic josamycin

(2009) Piotr Przybylski et al.   TETRAHEDRON LETTERS

Novel 16-membered macrolides modified at C-12 and C-13 positions of midecamycin A1 and miokamycin. Part 1: Synthesis and evaluation of 12,13-carbamate and 12-arylalkylamino-13-hydroxy analogues

(2008) Tomoaki Miura et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of novel leucomycin analogues modified at the C-3 position. Part II: 3-O-(3-Aryl-2-propenyl)leucomycin analogues

(2008) Takeshi Furuuchi et al.   BIOORGANIC & MEDICINAL CHEMISTRY