S8-Mediated Cyclization of 2-Aminophenols/thiophenols with Arylmethyl Chloride: Approach to Benzoxazoles and Benzothiazoles

Sulfur Containing Scaffolds in Drugs: Synthesis and Application in Medicinal Chemistry

(2016) Minghao Feng et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Sulphur promoted C(sp3)–C(sp2) cross dehydrogenative cyclisation of acetophenone hydrazones with aldehydes: efficient synthesis of 3,4,5-trisubstituted 1H-pyrazoles

(2015) Rajeshwer Vanjari et al.   CHEMICAL COMMUNICATIONS

Elemental Sulfur Mediated Decarboxylative Redox Cyclization Reaction of o-Chloronitroarenes and Arylacetic Acids

(2015) Tirumaleswararao Guntreddi et al.   ORGANIC LETTERS

Elemental Sulfur Disproportionation in the Redox Condensation Reaction betweeno-Halonitrobenzenes and Benzylamines

(2014) Thanh Binh Nguyen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A ball-milling strategy for the synthesis of benzothiazole, benzimidazole and benzoxazole derivatives under solvent-free conditions

(2014) Hemant Sharma et al.   GREEN CHEMISTRY

Decarboxylative Thioamidation of Arylacetic and Cinnamic Acids: A New Approach to Thioamides

(2014) Tirumaleswararao Guntreddi et al.   ORGANIC LETTERS

Copper-Catalyzed Synthesis of α-Trifluoromethylthio-Substituted Ketones

(2014) Yangjie Huang et al.   ORGANIC LETTERS

A simple approach to benzothiazoles from 2-chloronitrobenzene, elemental sulfur, and aliphatic amine under solvent-free and catalyst-free conditions

(2014) Yao Tong et al.   TETRAHEDRON LETTERS

Visible-Light-Mediated Decarboxylation/Oxidative Amidation of α-Keto Acids with Amines under Mild Reaction Conditions Using O2

(2013) Jie Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transfer of Sulfur: From Simple to Diverse

(2013) Hui Liu et al.   Chemistry-An Asian Journal

Palladium-Catalyzedortho-Aroylation of 2-Arylbenzothiazoles and 2-Arylbenzoxazoles with Aldehydes

(2013) Arghya Banerjee et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Oxidative Decarboxylative Arylation of Benzothiazoles with Phenylacetic Acids and α-Hydroxyphenylacetic Acids with O2 as the Sole Oxidant

(2013) Qiuling Song et al.   ORGANIC LETTERS

A Simple and Straightforward Approach to Quinoxalines by Iron/Sulfur-Catalyzed Redox Condensation of o-Nitroanilines and Phenethylamines

(2013) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Three-Component Reaction between Alkynes, Elemental Sulfur, and Aliphatic Amines: A General, Straightforward, and Atom Economical Approach to Thioamides

(2013) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Pd(PPh3)4-catalyzed direct ortho-fluorination of 2-arylbenzothiazoles with an electrophilic fluoride N-fluorobenzenesulfonimide (NFSI)

(2013) Qiuping Ding et al.   TETRAHEDRON

Cu-Catalyzed Three-Component Synthesis of Substituted Benzothiazoles in Water

(2012) Hang Deng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Iron Sulfide Catalyzed Redox/Condensation Cascade Reaction between 2-Amino/Hydroxy Nitrobenzenes and Activated Methyl Groups: A Straightforward Atom Economical Approach to 2-Hetaryl-benzimidazoles and -benzoxazoles

(2012) Thanh Binh Nguyen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Benzazoles from Aliphatic Amines and o-Amino/Mercaptan/Hydroxyanilines: Elemental Sulfur as a Highly Efficient and Traceless Oxidizing Agent

(2012) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Efficient and Selective Multicomponent Oxidative Coupling of Two Different Aliphatic Primary Amines into Thioamides by Elemental Sulfur

(2012) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Selection and Scale-Up Evaluation of an Alternative Route to (−)-(3R,4R)-1-Benzyl-4-(benzylamino)piperidin-3-ol

(2012) Ian S. Young et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Push–pull bithiophene azo-chromophores bearing thiazole and benzothiazole acceptor moieties: Synthesis and evaluation of their redox and nonlinear optical properties

(2011) M. Manuela M. Raposo et al.   DYES AND PIGMENTS

Difluoromethylbenzoxazole Pyrimidine Thioether Derivatives: A Novel Class of Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

(2011) Jérémie Boyer et al.   JOURNAL OF MEDICINAL CHEMISTRY

High regiocontrol in the nucleophilic ring opening of 1-aralkyl-3,4-epoxypiperidines with amines—a short-step synthesis of 4-fluorobenzyltrozamicol and novel anilidopiperidines

(2011) Matthias Scheunemann et al.   TETRAHEDRON

Copper-Catalyzed Intramolecular C−N Bond Formation: A Straightforward Synthesis of Benzimidazole Derivatives in Water

(2010) Jinsong Peng et al.   JOURNAL OF ORGANIC CHEMISTRY

Efficient and Economical Access to Substituted Benzothiazoles: Copper-Catalyzed Coupling of 2-Haloanilides with Metal Sulfides and Subsequent Condensation

(2009) Dawei Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

2-Arylbenzothiazole as a Privileged Scaffold in Drug Discovery

(2009) A. Weekes et al.   CURRENT MEDICINAL CHEMISTRY

Synthesis and Evaluation of18F-Labeled 2-Phenylbenzothiazoles as Positron Emission Tomography Imaging Agents for Amyloid Plaques in Alzheimer’s Disease

(2009) Kim Serdons et al.   JOURNAL OF MEDICINAL CHEMISTRY

Ligand-Free Copper-Catalyzed Synthesis of Substituted Benzimidazoles, 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and Benzoxazoles

(2009) Prasenjit Saha et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Biological Properties of Benzothiazole, Benzoxazole, and Chromen-4-one Analogues of the Potent Antitumor Agent 2-(3,4-Dimethoxyphenyl)-5-fluorobenzothiazole (PMX 610, NSC 721648)(1)

(2008) Stefania Aiello et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Synthesis of Benzimidazoles via Cascade Reactions ofo-Haloacetanilide Derivatives with Amidine Hydrochlorides

(2008) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis, metal ion binding, and biological evaluation of new anticancer 2-(2′-hydroxyphenyl)benzoxazole analogs of UK-1

(2007) Mireya L. McKee et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Biochemical and Structural Evaluation of Highly Selective 2-Arylbenzoxazole-Based Transthyretin Amyloidogenesis Inhibitors

(2007) Steven M. Johnson et al.   JOURNAL OF MEDICINAL CHEMISTRY