Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation

Rutaecarpine: A Promising Cardiovascular Protective Alkaloid from Evodia Rutaecarpa (Wu Zhu Yu)

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Multi-modal antidepressant-like action of 6- and 7-chloro-2-aminodihydroquinazolines in the mouse tail suspension test

(2019) Kavita A. Iyer et al.   PSYCHOPHARMACOLOGY

Anti-tubercular Potency and Computationallyassessed Drug-likeness and Toxicology of Diversely Substituted Indolizines

(2019) Katharigatta N Venugopala et al.   Indian Journal of Pharmaceutical Education and Research

Synthesis and insecticidal activity studies of novel phenylpyrazole derivatives containing arylimine or carbimidate moiety

(2019) Qiqi Zhao et al.   BIOORGANIC & MEDICINAL CHEMISTRY

2,4‐Diphenyl‐1,2‐dihydroquinazoline Derivatives: Synthesis, Anticancer Activity and Docking Studies

(2019) Krishna Kanthi Gudimella et al.   ChemistrySelect

Synthesis, Structural Studies, and α-Glucosidase Inhibitory, Antidiabetic, and Antioxidant Activities of 2,3-Dihydroquinazolin-4(1H)-ones Derived from Pyrazol-4-carbaldehyde and Anilines

(2019) Alireza Barmak et al.   ACS Omega

Anti-neuroinflammatory effects of tryptanthrin from Polygonum tinctorium Lour. in lipopolysaccharide-stimulated BV2 microglial cells

(2018) Seungjun Lee et al.   ARCHIVES OF PHARMACAL RESEARCH

Synthesis and Structural Elucidation of Novel 2,4-Disubstituted 1,3-Oxazole Analogues for Pharmacological Properties

(2018) Katharigatta N. Venugopala   ASIAN JOURNAL OF CHEMISTRY

Larvicidal study of tetrahydropyrimidine scaffolds against Anopheles arabiensis and structural insight by single crystal X-ray studies

(2018) Keshab M. Bairagi et al.   Chemical Biology & Drug Design

One-pot microwave assisted synthesis and structural elucidation of novel ethyl 3-substituted-7-methylindolizine-1-carboxylates with larvicidal activity against Anopheles arabiensis

(2018) Sandeep Chandrashekharappa et al.   JOURNAL OF MOLECULAR STRUCTURE

Efficient synthesis and characterization of novel indolizines: exploration of in vitro COX-2 inhibitory activity and molecular modelling studies

(2018) Sandeep Chandrashekharappa et al.   NEW JOURNAL OF CHEMISTRY

Structure of the G119S Mutant Acetylcholinesterase of the Malaria Vector Anopheles gambiae Reveals Basis of Insecticide Resistance

(2018) Jonah Cheung et al.   STRUCTURE

Noncovalent Inhibitors of Mosquito Acetylcholinesterase 1 with Resistance-Breaking Potency

(2018) Sofie Knutsson et al.   JOURNAL OF MEDICINAL CHEMISTRY

Crystal structure of acetylcholinesterase catalytic subunits of the malaria vector Anopheles gambiae

(2017) Qian Han et al.   Insect Science

A mosquito hemolymph odorant-binding protein family member specifically binds juvenile hormone

(2017) Il Hwan Kim et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Asymmetric Hydrogen Bonding Catalysis for the Synthesis of Dihydroquinazoline-Containing Antiviral, Letermovir

(2017) Cheol K. Chung et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Carbon–SO3H derived from glycerol: a green recyclable catalyst for synthesis of 2,3-dihydroquinazolin-4(1H)-ones

(2017) Rathinam Ramesh et al.   Journal of the Iranian Chemical Society

Synthesis and characterization of bromine source supported on magnetic Fe3 O4 nanoparticles: A new, versatile and efficient magnetically separable catalyst for organic synthesis

(2016) Lotfi Shiri et al.   APPLIED ORGANOMETALLIC CHEMISTRY

C ring may be dispensable for β-carboline: Design, synthesis, and bioactivities evaluation of tryptophan analog derivatives based on the biosynthesis of β-carboline alkaloids

(2016) Yuanqiong Huang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Greener synthesis of indolizine analogues using water as a base and solvent: study for larvicidal activity againstAnopheles arabiensis

(2016) Chandrashekharappa Sandeep et al.   Chemical Biology & Drug Design

Thiosemicarbazones as Aedes aegypti larvicidal

(2015) João Bosco P. da Silva et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Sulfonic acid functionalized Wang resin (Wang-OSO3H) as polymeric acidic catalyst for the eco-friendly synthesis of 2,3-dihydroquinazolin-4(1H)-ones

(2015) A.V. Dhanunjaya Rao et al.   TETRAHEDRON LETTERS

Efficient and green sulfamic acid catalyzed synthesis of new 1,2-dihydroquinazoline derivatives with antibacterial potential

(2015) Ahmed Kamal et al.   Arabian Journal of Chemistry

PLATONSQUEEZE: a tool for the calculation of the disordered solvent contribution to the calculated structure factors

(2015) Anthony L. Spek   Acta Crystallographica Section C-Structural Chemistry

Crystal structure refinement withSHELXL

(2015) George M. Sheldrick   Acta Crystallographica Section C-Structural Chemistry

Synthesis of novel thiadiazolotriazin-4-ones and study of their mosquito-larvicidal and antibacterial properties

(2014) Prakash Anil Castelino et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Development of potent and selective Plasmodium falciparum calcium-dependent protein kinase 4 (PfCDPK4) inhibitors that block the transmission of malaria to mosquitoes

(2014) Rama Subba Rao Vidadala et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Antimosquito Properties of 2-Substituted Phenyl/benzylamino-6-(4- chlorophenyl)-5-methoxycarbonyl-4-methyl-3,6-dihydropyrimidin-1-ium Chlorides Against Anopheles arabiensis

(2014) Venugopala Narayanaswamy et al.   Medicinal Chemistry

Insecticide resistance in Anopheles arabiensis in Sudan: temporal trends and underlying mechanisms

(2014) Hiba Abdalla et al.   Parasites & Vectors

The enzyme 3-hydroxykynurenine transaminase as potential target for 1,2,4-oxadiazoles with larvicide activity against the dengue vector Aedes aegypti

(2013) Vanessa S. Oliveira et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and insecticidal activities of 2,3-dihydroquinazolin-4(1H)-one derivatives targeting calcium channel

(2013) Yunyun Zhou et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and antimosquito properties of 2,6-substituted benzo[d]thiazole and 2,4-substituted benzo[d]thiazole analogues against Anopheles arabiensis

(2013) Katharigatta Narayanaswamy Venugopala et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Fungicidal Activity, and Sterol 14α-Demethylase Binding Interaction of 2-Azolyl-3,4-dihydroquinazolines on Penicillium digitatum

(2013) Wen-Jin Li et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Synthesis and characterization of quinazoline derivatives: search for hybrid molecule as diuretic and antihypertensive agents

(2013) Mujeeb Ur Rahman et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Synthesis, antibacterial and antioxidant activity of novel 2,3-dihydroquinazolin-4(1H)-one derivatives of dehydroabietylamine diterpene

(2013) Peyman Salehi et al.   Journal of the Iranian Chemical Society

The global distribution and burden of dengue

(2013) Samir Bhatt et al.   NATURE

Discovery of a Novel Broad-Spectrum Antifungal Agent Derived from Albaconazole

(2013) Rémi Guillon et al.   ACS Medicinal Chemistry Letters

Synthesis and insecticidal evaluation of novel N-pyridylpyrazolecarboxamides containing cyano substituent in the ortho-position

(2012) Mingzhen Mao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

WinGXandORTEP for Windows: an update

(2012) Louis J. Farrugia   JOURNAL OF APPLIED CRYSTALLOGRAPHY

Molecular docking and receptor-specific 3D-QSAR studies of acetylcholinesterase inhibitors

(2012) Pran Kishore Deb et al.   MOLECULAR DIVERSITY

New conditions for synthesis of (±)-2-monosubstituted and (±)-2,2-disubstituted 2,3-dihydro-4(1H)-quinazolinones from 2-nitro- and 2-aminobenzamide

(2011) Richard A. Bunce et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Recent Advances in the Studies on Luotonins

(2011) Jing Lu Liang et al.   MOLECULES

Synthesis of New 2,3-Dihydroquinazolin-4(1H)-one Derivatives for Analgesic and Anti-inflammatory Evaluation

(2010) Osama I. El-Sabbagh et al.   ARCHIV DER PHARMAZIE

Microwave-induced synthesis of schiff bases of aminothiazolyl bromocoumarins as antibacterials

(2009) KN Venugopala et al.   INDIAN JOURNAL OF PHARMACEUTICAL SCIENCES