Substrate or Solvent-Controlled PdII -Catalyzed Regioselective Arylation of Quinolin-4(1H )-ones Using Diaryliodonium Salts: Facile Access to Benzoxocine and Aaptamine Analogues

Cobalt-Catalyzed C−H Nitration of Indoles by Employing a Removable Directing Group

(2018) Paridhi Saxena et al.   Chemistry-An Asian Journal

Transient Directing Groups for Transformative C–H Activation by Synergistic Metal Catalysis

(2018) Parthasarathy Gandeepan et al.   Chem

Enhanced Reactivity by Torsional Strain of Cyclic Diaryliodonium in Cu-Catalyzed Enantioselective Ring-Opening Reaction

(2018) Kun Zhao et al.   Chem

Copper-Catalyzed Asymmetric Ring-Opening of Cyclic Diaryliodonium with Benzylic and Aliphatic Amines

(2018) Shibo Xu et al.   ADVANCED SYNTHESIS & CATALYSIS

A comprehensive overview of directing groups applied in metal-catalysed C–H functionalisation chemistry

(2018) Carlo Sambiagio et al.   CHEMICAL SOCIETY REVIEWS

Synthesis and Application of Cyclic Diaryliodonium Salts: A Platform for Bifunctionalization in a Single Step

(2017) Nachiketa Chatterjee et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Thieno-Fused Five- and Six-Membered Nitrogen and Oxygen Heterocycles via Intramolecular Heteroannulation of 4,5-Substituted 3-Amino or 3-Hydroxy 2-Functionalized Thiophenes

(2017) Anand Acharya et al.   JOURNAL OF ORGANIC CHEMISTRY

Substrate-Controlled Regioselective Arylations of 2-Indolylmethanols with Indoles: Synthesis of Bis(indolyl)methane and 3,3′-Bisindole Derivatives

(2017) Ying-Ying He et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed, ortho-Selective C–H Halogenation of Benzyl Nitriles, Aryl Weinreb Amides, and Anilides

(2017) Riki Das et al.   JOURNAL OF ORGANIC CHEMISTRY

Diverse ortho-C(sp2)–H Functionalization of Benzaldehydes Using Transient Directing Groups

(2017) Xi-Hai Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regioselective access of alkylidendibenzo[c,f]oxocine framework via cyclocarbopalladation/cross-coupling cascade reactions and reductive Heck strategy

(2017) Tapas Ghosh   NEW JOURNAL OF CHEMISTRY

Pd-Catalyzed Direct ortho-C–H Arylation of Aromatic Ketones Enabled by a Transient Directing Group

(2017) Jiancong Xu et al.   ORGANIC LETTERS

Electrophilic Ring Opening of Small Heterocycles

(2017) Chuan Wang   SYNTHESIS-STUTTGART

A Simple and Versatile Amide Directing Group for C−H Functionalizations

(2016) Ru-Yi Zhu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Advances in Synthetic Applications of Hypervalent Iodine Compounds

(2016) Akira Yoshimura et al.   CHEMICAL REVIEWS

Pd-Catalyzed Ligand-Free Synthesis of Arylated Heteroaromatics by Coupling of N-Heteroaromatic Bromides with Iodobenzene Diacetate, Iodosobenzene, or Diphenyliodonium Salts

(2016) Xiajun Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

One Substrate, Two Modes of C–H Functionalization: A Metal-Controlled Site-Selectivity Switch in C–H Arylation Reactions

(2016) Virendra Kumar Tiwari et al.   ORGANIC LETTERS

Acetohydrazone: A Transient Directing Group for Arylation of Unactivated C(sp3)–H Bonds

(2016) Fei Ma et al.   ORGANIC LETTERS

Palladium(II)-Catalyzed, Heteroatom-Directed, Regioselective C–H Nitration of Anilines Using Pyrimidine as a Removable Directing Group

(2016) Govind Goroba Pawar et al.   ORGANIC LETTERS

Functionalization of C(sp3)-H bonds using a transient directing group

(2016) F.-L. Zhang et al.   SCIENCE

Diaryliodonium Salts in Organic Syntheses: A Useful Compound Class for Novel Arylation Strategies

(2016) Zoltán Novák et al.   SYNLETT

β-Arylation of oxime ethers using diaryliodonium salts through activation of inert C(sp)–H bonds using a palladium catalyst

(2016) Jing Peng et al.   Chemical Science

Synthesis of isocryptolepine analogues and their structure–activity relationship studies as antiplasmodial and antiproliferative agents

(2015) Pasuk Aroonkit et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Ohmic Heating-Assisted Synthesis of 3-Arylquinolin-4(1H)-ones by a Reusable and Ligand-Free Suzuki–Miyaura Reaction in Water

(2015) Joana Pinto et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalyst Controlled Divergent C4/C8 Site-Selective C–H Arylation of Isoquinolones

(2015) Soyoung Lee et al.   ORGANIC LETTERS

Gold-Catalyzed 1,2-Acyloxy Migration/Intramolecular [3+2] 1,3-Dipolar Cycloaddtion Cascade Reaction: An Efficient Strategy for Syntheses of Medium-Sized-Ring Ethers and Amines

(2014) Changgui Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of (±)-Distomadines A and B

(2014) Alexandre E. R. Jolibois et al.   ORGANIC LETTERS

Recent advances in directed C–H functionalizations using monodentate nitrogen-based directing groups

(2014) Min Zhang et al.   Organic Chemistry Frontiers

Palladium-Catalyzedortho-Selective CH Deuteration of Arenes: Evidence for Superior Reactivity of Weakly Coordinated Palladacycles

(2013) Sandy Ma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cu-Catalyzed Fluorination of Diaryliodonium Salts with KF

(2013) Naoko Ichiishi et al.   ORGANIC LETTERS

Lead Optimization of 3-Carboxyl-4(1H)-Quinolones to Deliver Orally Bioavailable Antimalarials

(2012) Yiqun Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Palladium-Catalyzed Decarboxylative Coupling of Quinolinone-3-Carboxylic Acids and Related Heterocyclic Carboxylic Acids with (Hetero)aryl Halides

(2012) Samir Messaoudi et al.   ORGANIC LETTERS

Gold(I)-Catalyzed Synthesis of Benzoxocines by an 8-endo-dig Cyclization

(2011) Kathrin Wittstein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and antimalarial evaluation of novel isocryptolepine derivatives

(2011) Louise R. Whittell et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and antiproliferative evaluation of certain indolo[3,2-c]quinoline derivatives

(2010) Chih-Ming Lu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Effects of haloniums on gold-catalyzed ring expansion of 1-oxiranyl-1-alkynylcyclopropanes

(2010) Hsuan-Hung Liao et al.   CHEMICAL COMMUNICATIONS

Antimalarial Activity of Novel 5-Aryl-8-Aminoquinoline Derivatives

(2010) Hiroaki Shiraki et al.   JOURNAL OF MEDICINAL CHEMISTRY

Diaryliodonium Salts: A Journey from Obscurity to Fame

(2009) Eleanor���A. Merritt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and structure–activity relationships of cassiarin A as potential antimalarials with vasorelaxant activity

(2009) Hiroshi Morita et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Aaptamine and related products. Their isolation, chemical syntheses, and biological activity

(2009) Enrique L. Larghi et al.   TETRAHEDRON

A formal total synthesis of the marine alkaloid aaptamine

(2008) Enrique L. Larghi et al.   TETRAHEDRON