2-Bromo-2-chloro-3-arylpropanenitriles as C-3 Synthons for the Synthesis of Functionalized 3-Aminothiophenes

Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors

(2019) Romeo Romagnoli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Straightforward Synthesis of 3‐Aminothiophenes Using Activated Amides

(2019) Dylan Dagoneau et al.   HELVETICA CHIMICA ACTA

Pluripotent Features of Doubly Thiophene‐Fused Benzodiphospholes as Organic Functional Materials

(2019) Tomohiro Higashino et al.   CHEMISTRY-A EUROPEAN JOURNAL

Thiophenes from Echinops grijsii as a Preliminary Approach To Control Disease Complex of Root-Knot Nematodes and Soil-Borne Fungi: Isolation, Activities, and Structure–Nonphototoxic Activity Relationship Analysis

(2019) Tingting Liu et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

New Chalcone Derivatives with Schiff Base-Thiophene: Synthesis, Biological Activity, and Molecular Docking Studies

(2019) Y. Ünver et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Improved one-pot synthetic conditions for synthesis of functionalized fluorescent coumarin-thiophene hybrids: Syntheses, DFT studies, photophysical and thermal properties

(2019) Issah Yahaya et al.   TETRAHEDRON

Nonlinear Nonacenes with a Dithienothiophene Substructure: Multifunctional Compounds that Act as Columnar Mesogens, Luminophores, π Gelators, and p‐Type Semiconductors

(2019) Tao Ma et al.   ChemPlusChem

5-Nitro-Thiophene-Thiosemicarbazone Derivatives Present Antitumor Activity Mediated by Apoptosis and DNA Intercalation

(2019) Karla Mirella Roque Marques et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Synthesis of New Derivatives of 4-(1,4-Benzodioxan-2-yl)thiophene

(2019) S. O. Vardanyan et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Anticancer Activity of Thiophene-2-carboxamide Derivatives and In Silico Docking Studies

(2019) K. C. Gulipalli et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Synthesis of Some New Substituted Thieno[2,3-d]pyrimidine Derivatives as Antimicrobial Agents

(2019) M. F. El-Shehry et al.   RUSSIAN JOURNAL OF GENERAL CHEMISTRY

Design and synthesis of novel 3-(thiophen-2-yl)-1,5-dihydro-2H-pyrrol-2-one derivatives bearing a hydrazone moiety as potential fungicides

(2018) Xiaobin Wang et al.   Chemistry Central Journal

2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition

(2018) Romeo Romagnoli et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Understanding the tetrazole ring cleavage reaction with hydrazines: Structural determination and mechanistic insight

(2018) Olga Ya. Shyyka et al.   TETRAHEDRON LETTERS

Synthetic Applications and Biological Properties of 1,4-Dithiane-2,5-diol and its Aducts: A Review

(2018) Isadora Silva Luna et al.   CURRENT ORGANIC SYNTHESIS

Therapeutic importance of synthetic thiophene

(2018) Rashmi Shah et al.   Chemistry Central Journal

3-Aryl Substituted 1-Methylquinolinium Salts as Carbene Precursors

(2018) Sviatoslav Batsyts et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis, Molecular Engineering, and Photophysical Properties of Fluorescent Thieno[3,2-b]pyridine-5(4H)-ones

(2018) Dan-Bi Sung et al.   JOURNAL OF ORGANIC CHEMISTRY

On the structure of transition metals complexes with the new tridentate dye of thiazole series: Theoretical and experimental studies

(2017) Maksym Fizer et al.   JOURNAL OF MOLECULAR STRUCTURE

Design, Synthesis and Anti-Proliferative Activities of 2,6-Substituted Thieno[3,2-d]pyrimidine Derivatives Containing Electrophilic Warheads

(2017) Qiumeng Zhang et al.   MOLECULES

Synthesis of [4-amino-5-(R-benzyl)-1,3-thiazol-2-ylsulfanyl] acetic acids

(2017) Yu. V. Ostapyuk et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Suzuki–Miyaura Cross-Coupling Reactions in Acetic Acid Employing Sydnone-Derived Catalyst Systems

(2017) Andreas Schmidt et al.   SYNLETT

N-Propargylic β-enaminocarbonyls: powerful and versatile building blocks in organic synthesis

(2017) Sattar Arshadi et al.   RSC Advances

An Aromatic Diamidine That Targets Kinetoplast DNA, Impairs the Cell Cycle in Trypanosoma cruzi, and Diminishes Trypomastigote Release from Infected Mammalian Host Cells

(2016) Richard M. B. M. Girard et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Dipolar Bent and Linear Acetylenes Substituted by Cationic Quinolinium and Anionic Benzoates. Formation of Mesomeric Betaines

(2016) Andreas Schmidt et al.   JOURNAL OF ORGANIC CHEMISTRY

Regio- and Stereoselective Cyanotriflation of Alkynes Using Aryl(cyano)iodonium Triflates

(2016) Xi Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent Advances in Meerwein Arylation Chemistry

(2016) Markus Heinrich et al.   SYNTHESIS-STUTTGART

A simple and convenient synthesis of 3-arylpyran-2-ones via the Meerwein reaction

(2016) Roman Z. Lytvyn et al.   TETRAHEDRON LETTERS

Palladium complexes of anionic N-heterocyclic carbenes derived from sydnones in catalysis

(2016) Ana-Luiza Lücke et al.   ZEITSCHRIFT FUR NATURFORSCHUNG SECTION B-A JOURNAL OF CHEMICAL SCIENCES

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium

(2015) Anita Cohen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Exploring the chemical space of ureidothiophene-2-carboxylic acids as inhibitors of the quorum sensing enzyme PqsD from Pseudomonas aeruginosa

(2015) J. Henning Sahner et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

How the Structural Elucidation of the Natural Product Stephanosporin Led to New Developments in Aryl Radical and Medicinal Chemistry

(2015) Markus Heinrich et al.   SYNLETT

New Convenient Strategy for Annulation of Pyrimidines to Thiophenes or Furans via the One-pot Multistep Cascade Reaction of 1H-Tetrazoles with Aliphatic Amines

(2015) Nazariy T. Pokhodylo et al.   ACS Combinatorial Science

Crystal structure refinement withSHELXL

(2015) George M. Sheldrick   Acta Crystallographica Section C-Structural Chemistry

Synthesis of 3-Aryl/methoxycarbonyl-3,4-dihydroisocoumarin-6-carboxylic Acid Derivatives

(2014) Victor V. Turytsya et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Graphene based material as a base catalyst for solvent free Aldol condensation and Knoevenagel reaction at room temperature

(2014) Sk Manirul Islam et al.   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Novel small molecule inhibitors targeting the “switch region” of bacterial RNAP: Structure-based optimization of a virtual screening hit

(2013) J. Henning Sahner et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Organometallic Schiff bases derived from 5-nitrothiophene and 5-nitrofurane: Synthesis, crystallographic, electrochemical, ESR and antiTrypanosoma cruzi studies

(2013) Rodrigo Arancibia et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Facile and Efficient One-Pot Procedure for Thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines Preparation

(2013) Nazariy T. Pokhodylo et al.   SYNTHETIC COMMUNICATIONS

Development of Novel Alkene Oxindole Derivatives As Orally Efficacious AMP-Activated Protein Kinase Activators

(2013) Li-Fang Yu et al.   ACS Medicinal Chemistry Letters

Convenient synthesis of α-bromo ketones by the Meerwein reaction

(2012) Yu. V. Ostapiuk et al.   RUSSIAN JOURNAL OF ORGANIC CHEMISTRY

Photocatalytic Arylation of Alkenes, Alkynes and Enones with Diazonium Salts

(2012) Peter Schroll et al.   ChemistryOpen

Selective Mono- to Perarylations of Tetrabromothiophene by a Cyclobutene-1,2-diylbisimidazolium Preligand

(2011) Alireza Rahimi et al.   JOURNAL OF ORGANIC CHEMISTRY

A convenient method for the synthesis of 2-[(5-benzyl-1,3-thiazol-2-yl)imino]-1,3-thiazolidin-4-one derivatives

(2011) Yuri V. Ostapiuk et al.   TETRAHEDRON LETTERS

Gallium (iii)-catalysed bromocyanation of alkynes: regio- and stereoselective synthesis of β-bromo-α,β-unsaturated nitriles

(2010) Masahito Murai et al.   CHEMICAL COMMUNICATIONS

Synthesis of heterocycles on the basis of products of arylation of unsaturated compounds 22.* 3-Aryl-2-chloropropanal in the synthesis of N-Aryl-5-(R-benzyl)-1,3-thiazole-2-amines

(2010) V. S. Matiychuk et al.   Chemistry of Heterocyclic Compounds

Bicyclic Substituted Hydroxyphenylmethanones as Novel Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 1 (17β-HSD1) for the Treatment of Estrogen-Dependent Diseases

(2010) Alexander Oster et al.   JOURNAL OF MEDICINAL CHEMISTRY

Three-component condensation of 3-aminothiophene-2-carboxylic acid derivatives with aldehydes and Meldrum’s acid

(2010) B. V. Lichitsky et al.   RUSSIAN CHEMICAL BULLETIN

OLEX2: a complete structure solution, refinement and analysis program

(2009) Oleg V. Dolomanov et al.   JOURNAL OF APPLIED CRYSTALLOGRAPHY

Synthesis of ethyl 4,5-disubstituted 2-azido-3-thiophenecarboxylates and use in the synthesis of thieno[3,2-e][1,2,3]triazolo[1,5-a]pyrimidin-5(4H)-ones

(2009) Nazariy T. Pokhodylo et al.   TETRAHEDRON

Intermolecular Olefin Functionalisation Involving Aryl Radicals Generated from Arenediazonium Salts

(2008) Markus R. Heinrich   CHEMISTRY-A EUROPEAN JOURNAL

Design, Synthesis, Biological Evaluation and Pharmacokinetics of Bis(hydroxyphenyl) substituted Azoles, Thiophenes, Benzenes, and Aza-Benzenes as Potent and Selective Nonsteroidal Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 1 (17β-HSD1)

(2008) Emmanuel Bey et al.   JOURNAL OF MEDICINAL CHEMISTRY

Theoretical Study on Structural, Electronic, and Optical Properties of Ambipolar Diphenylamino End-capped Oligofluorenylthiophenes and Fluoroarene-thiophene as Light-emitting Materials

(2008) Xue-Qin Ran et al.   JOURNAL OF PHYSICAL CHEMISTRY A

One-pot synthesis of substituted 3-amino-2-nitrothiophenes and selenophenes

(2008) David Thomae et al.   TETRAHEDRON