Targeting epigenetic reader and eraser: Rational design, synthesis and in vitro evaluation of dimethylisoxazoles derivatives as BRD4/HDAC dual inhibitors

Title
Targeting epigenetic reader and eraser: Rational design, synthesis and in vitro evaluation of dimethylisoxazoles derivatives as BRD4/HDAC dual inhibitors
Authors
Keywords
Epigenetic, Protein–protein interactions, Bromodomain, HDAC, Antiproliferative activity
Journal
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Volume 26, Issue 12, Pages 2931-2935
Publisher
Elsevier BV
Online
2016-04-29
DOI
10.1016/j.bmcl.2016.04.034

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