Journal
CHINESE CHEMICAL LETTERS
Volume 31, Issue 5, Pages 1332-1336Publisher
ELSEVIER SCIENCE INC
DOI: 10.1016/j.cclet.2019.10.035
Keywords
Indole; Diastereoselective; Dearomatization; 2,3-Diazidation; Indoline
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Funding
- National Natural Science Foundation of China [21472172, 21272212]
- Natural Science Foundation of Zhejiang Province [LY17B060009]
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The copper-catalyzed directed dearomatization of indoles with the assistance of directing groups has been developed for the synthesis of 2,3-diazido indolines with good yields and excellent diastereoselectivities in aqueous solution. The resultant 2,3-diazides can be smoothly converted to other functional groups, including vicinal diamines, triazoles and benzotriazoles, in a single step. (C) 2019 Chinese Chemical Society and Institute of Materia Medica, Chinese Academy of Medical Sciences. Published by Elsevier B.V. All rights reserved.
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