Chemical synthesis, molecular modeling and pharmacophore mapping of new pyrrole derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth

Synthesis, biological evaluation and in silico molecular modeling of pyrrolyl benzohydrazide derivatives as enoyl ACP reductase inhibitors

(2017) Shrinivas D. Joshi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

N-Benzyl-4-((heteroaryl)methyl)benzamides: A New Class of Direct NADH-Dependent 2-transEnoyl-Acyl Carrier Protein Reductase (InhA) Inhibitors with Antitubercular Activity

(2016) Ana Guardia et al.   ChemMedChem

Synthesis, characterization and antitubercular activities of novel pyrrolyl hydrazones and their Cu-complexes

(2016) Shrinivas D. Joshi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Drug Resistance of Antitubercular Agents at the Genetic Level in Mycobacterium Species: A Road Map to Drug Development for Counteracting the Resistance

(2016) Shrinivas D. Joshi et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth

(2015) Aurélien Chollet et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Enoyl ACP Reductase as Effective Target for the Synthesized Novel Antitubercular Drugs: A-State-of-the-Art

(2014) Shrinivas Joshi et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents

(2012) Christophe Menendez et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis of some new (2-aminothiazol-4-yl)methylester derivatives as possible antimicrobial and antitubercular agents

(2012) Ranjith P. Karuvalam et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological activities of triazole derivatives as inhibitors of InhA and antituberculosis agents

(2011) Christophe Menendez et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Ligand-based pharmacophore model of N-Aryl and N-Heteroaryl piperazine α1A-adrenoceptors antagonists using GALAHAD

(2010) Xin Zhao et al.   JOURNAL OF MOLECULAR GRAPHICS & MODELLING

3D-QSAR (CoMFA and CoMSIA) and pharmacophore (GALAHAD) studies on the differential inhibition of aldose reductase by flavonoid compounds

(2010) Julio Caballero   JOURNAL OF MOLECULAR GRAPHICS & MODELLING

Synthesis of new 4-pyrrol-1-yl benzoic acid hydrazide analogs and some derived oxadiazole, triazole and pyrrole ring systems: A novel class of potential antibacterial and antitubercular agents

(2007) S.D. Joshi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY