Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino)pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies

Title
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino)pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies
Authors
Keywords
CHK1 kinase inhibitor, Selectivity, Monotherapy, Hematologic malignancies
Journal
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 173, Issue -, Pages 44-62
Publisher
Elsevier BV
Online
2019-04-03
DOI
10.1016/j.ejmech.2019.03.062

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