Transition‐Metal‐Free Aryl–Aryl Cross‐Coupling: C−H Arylation of 2‐Naphthols with Diaryliodonium Salts

Transition-Metal-Free Desulfinative Cross-Coupling of Heteroaryl Sulfinates with Grignard Reagents

(2019) Jun Wei et al.   ORGANIC LETTERS

Metal-Free Synthesis of Pharmaceutically Important Biaryls by Photosplicing

(2018) Florian Kloss et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Sigmatropic Rearrangements of Hypervalent-Iodine-Tethered Intermediates for the Synthesis of Biaryls

(2018) Mitsuki Hori et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral phosphoric acid catalysis: from numbers to insights

(2018) Rajat Maji et al.   CHEMICAL SOCIETY REVIEWS

Transition-Metal-Free Suzuki-Type Cross-Coupling Reaction of Benzyl Halides and Boronic Acids via 1,2-Metalate Shift

(2018) Zhiqi He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Selective, Catalytic, and Metal-Free Coupling of Electron-Rich Phenols and Anilides Using Molecular Oxygen as Terminal Oxidant

(2018) Luis Bering et al.   ORGANIC LETTERS

Transition Metal-free Approaches to Biaryls

(2018) Francesca Piazzolla et al.   CURRENT ORGANIC CHEMISTRY

Heterobiaryl synthesis by contractive C–C coupling via P(V) intermediates

(2018) Michael C. Hilton et al.   SCIENCE

Oxidative Cross-Coupling of Substituted Phenols with Unactivated Aromatics

(2017) Nagnath Yadav More et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Oxidative Biaryl Coupling of N-Aryl Anilines by Using a Hypervalent Iodine(III) Reagent

(2017) Yasuyuki Kita et al.   SYNLETT

Metal-free Oxidative Cross-Coupling Reaction of Aromatic Compounds Containing Heteroatoms

(2017) Yasuyuki Kita et al.   SYNLETT

P(NMe 2 ) 3 -promoted ortho -selective arylation of phenols with diaryliodonium triflates via rhodium catalysis

(2017) Qi-Sheng Liu et al.   TETRAHEDRON

Regioselective synthesis of C3 alkylated and arylated benzothiophenes

(2017) Harry J. Shrives et al.   Nature Communications

Organo-Iodine(III)-Catalyzed Oxidative Phenol-Arene and Phenol-Phenol Cross-Coupling Reaction

(2016) Koji Morimoto et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal Free Bi(hetero)aryl Synthesis: A Benzyne Truce-Smiles Rearrangement

(2016) Catherine M. Holden et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Quinine-Catalyzed Asymmetric Synthesis of 2,2′-Binaphthol-Type Biaryls under Mild Reaction Conditions

(2016) Mauro Moliterno et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient Coupling Reaction of Quinone Monoacetal with Phenols Leading to Phenol Biaryls

(2016) Tohru Kamitanaka et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas

(2016) Yu Zhou et al.   CHEMICAL REVIEWS

Metal-Free Approach to Biaryls from Phenols and Aryl Sulfoxides by Temporarily Sulfur-Tethered Regioselective C–H/C–H Coupling

(2016) Tomoyuki Yanagi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Symmetry in Cascade Chirality-Transfer Processes: A Catalytic Atroposelective Direct Arylation Approach to BINOL Derivatives

(2016) Jin-Zheng Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric dearomatization of phenols

(2016) Wangsheng Sun et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-catalyzed selective ortho-arylations of 2-naphthol and phenol derivatives with diaryliodonium salts

(2016) Xiaofei Qian et al.   TETRAHEDRON LETTERS

Practical Organocatalytic Synthesis of Functionalized Non-C 2 -Symmetrical Atropisomeric Biaryls

(2015) Hongyin Gao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free Oxidative CC Bond Formation through CH Bond Functionalization

(2015) Rishikesh Narayan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Source of Selectivity in Oxidative Cross-Coupling of Aryls by Solvent Effect of 1,1,1,3,3,3-Hexafluoropropan-2-ol

(2015) Bernd Elsler et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fluorination Patterning: A Study of Structural Motifs That Impact Physicochemical Properties of Relevance to Drug Discovery

(2015) Quentin A. Huchet et al.   JOURNAL OF MEDICINAL CHEMISTRY

Applications of Fluorine in Medicinal Chemistry

(2015) Eric P. Gillis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Analysis of Past and Present Synthetic Methodologies on Medicinal Chemistry: Where Have All the New Reactions Gone?

(2015) Dean G. Brown et al.   JOURNAL OF MEDICINAL CHEMISTRY

Atroposelective Synthesis of Axially Chiral Biaryldiols via Organocatalytic Arylation of 2-Naphthols

(2015) Ye-Hui Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A counteranion triggered arylation strategy using diaryliodonium fluorides

(2015) L. Chan et al.   Chemical Science

The Biocatalytic Repertoire of Natural Biaryl Formation

(2014) Hülya Aldemir et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Free Coupling Reactions

(2014) Chang-Liang Sun et al.   CHEMICAL REVIEWS

Complete Field Guide to Asymmetric BINOL-Phosphate Derived Brønsted Acid and Metal Catalysis: History and Classification by Mode of Activation; Brønsted Acidity, Hydrogen Bonding, Ion Pairing, and Metal Phosphates

(2014) Dixit Parmar et al.   CHEMICAL REVIEWS

Comparison of Oxidative Aromatic Coupling and the Scholl Reaction

(2013) Marek Grzybowski et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free OxidativeparaCross-Coupling of Phenols

(2013) Koji Morimoto et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic C–H/C–H′ Cross-Biaryl Coupling: C-Selective Arylation of Sulfonanilides with Aromatic Hydrocarbons

(2013) Motoki Ito et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bioactive natural products derived from the Central African flora against neglected tropical diseases and HIV

(2013) Denis Zofou et al.   NATURAL PRODUCT REPORTS

Pyrene-cored blue-light emitting [4]helicenes: synthesis, crystal structures, and photophysical properties

(2013) Jian-Yong Hu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Metal-Free Synthesis of Aryl Ethers in Water

(2013) Erik Lindstedt et al.   ORGANIC LETTERS

Metal-Free Arylation of Oxygen Nucleophiles with Diaryliodonium Salts

(2012) Nazli Jalalian et al.   CHEMISTRY-A EUROPEAN JOURNAL

Efficient Anodic and Direct Phenol-Arene C,C Cross-Coupling: The Benign Role of Water or Methanol

(2012) Axel Kirste et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates

(2011) Stephen D. Roughley et al.   JOURNAL OF MEDICINAL CHEMISTRY

Room Temperature, Metal-Free Synthesis of Diaryl Ethers with Use of Diaryliodonium Salts

(2011) Nazli Jalalian et al.   ORGANIC LETTERS

α-Arylation by Rearrangement: On the Reaction of Enolates with Diaryliodonium Salts

(2010) Per-Ola Norrby et al.   CHEMISTRY-A EUROPEAN JOURNAL

Hypervalent iodine-mediated phenol dearomatization in natural product synthesis

(2010) Laurent Pouységu et al.   TETRAHEDRON

Anodic Phenol-Arene Cross-Coupling Reaction on Boron-Doped Diamond Electrodes

(2009) Axel Kirste et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION