First-generation structure-activity relationship studies of 2,3,4,9-tetrahydro-1H-carbazol-1-amines as CpxA phosphatase inhibitors

Title
First-generation structure-activity relationship studies of 2,3,4,9-tetrahydro-1H-carbazol-1-amines as CpxA phosphatase inhibitors
Authors
Keywords
Two-component system, Sensory kinase, Antibacterial, Drug discovery, Medicinal chemistry, CpxRA, Permeability, Efflux
Journal
Publisher
Elsevier BV
Online
2019-05-09
DOI
10.1016/j.bmcl.2019.05.003

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