Synthesis and biological evaluation of 1,2,4-oxadiazole linked 1,3,4-oxadiazole derivatives as tubulin binding agents

The MM/PBSA and MM/GBSA methods to estimate ligand-binding affinities

(2015) Samuel Genheden et al.   Expert Opinion on Drug Discovery

Zibotentan

(2015) N.D. James et al.   DRUGS OF THE FUTURE

A Conformational Mimetic Approach for the Synthesis of Carbocyclic Nucleosides as Anti-HCV Leads

(2013) Mohan Kasula et al.   ChemMedChem

Structure based medicinal chemistry approach to develop 4-methyl-7-deazaadenine carbocyclic nucleosides as anti-HCV agent

(2012) Anandarajan Thiyagarajan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Aromatic interaction profile to understand the molecular basis of raltegravir resistance

(2012) Tuniki Balaraju et al.   STRUCTURAL CHEMISTRY

Structure and Cytotoxicity of Phidianidines A and B: First Finding of 1,2,4-Oxadiazole System in a Marine Natural Product

(2011) Marianna Carbone et al.   ORGANIC LETTERS

The VSGB 2.0 model: A next generation energy model for high resolution protein structure modeling

(2011) Jianing Li et al.   PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS

Synthesis, characterization, and in vitro antimicrobial activities of 5-alkenyl/hydroxyalkenyl-2-phenylamine-1,3,4-oxadiazoles and thiadiazoles

(2010) Nida N. Farshori et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Convenient synthesis and biological profile of 5-amino-substituted 1,2,4-oxadiazole derivatives

(2010) Maria Ispikoudi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Discovery of a Long-Acting, Peripherally Selective Inhibitor of Catechol-O-methyltransferase

(2010) László E. Kiss et al.   JOURNAL OF MEDICINAL CHEMISTRY

Tuned methods for conjugate addition to a vinyl oxadiazole; synthesis of pharmaceutically important motifs

(2010) Alan R. Burns et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of novel 1,3,4-oxadiazole derivatives and their biological properties

(2009) Asif Husain et al.   ACTA PHARMACEUTICA

Design, synthesis and cruzain docking of 3-(4-substituted-aryl)-1,2,4-oxadiazole-N-acylhydrazones as anti-Trypanosoma cruzi agents

(2009) José Mauricio dos Santos Filho et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and pharmacological evaluation of 1,3,4-oxadiazole bearing bis(heterocycle) derivatives as anti-inflammatory and analgesic agents

(2009) B. Jayashankar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY