A bright future for fragment-based drug discovery: what does it hold?
Published 2019 View Full Article
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Title
A bright future for fragment-based drug discovery: what does it hold?
Authors
Keywords
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Journal
Expert Opinion on Drug Discovery
Volume -, Issue -, Pages 1-4
Publisher
Informa UK Limited
Online
2019-02-22
DOI
10.1080/17460441.2019.1583643
References
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- (2017) Bas Lamoree et al. Essays in Biochemistry
- Correction to When Does Chemical Elaboration Induce a Ligand To Change Its Binding Mode?
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- Design Principles for Fragment Libraries: Maximizing the Value of Learnings from Pharma Fragment-Based Drug Discovery (FBDD) Programs for Use in Academia
- (2016) György M. Keserű et al. JOURNAL OF MEDICINAL CHEMISTRY
- Identifying Interactions that Determine Fragment Binding at Protein Hotspots
- (2016) Chris J. Radoux et al. JOURNAL OF MEDICINAL CHEMISTRY
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- Twenty years on: the impact of fragments on drug discovery
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- Considerations of Protein Subpockets in Fragment-Based Drug Design
- (2015) Matthew Bartolowits et al. Chemical Biology & Drug Design
- Detection of secondary binding sites in proteins using fragment screening
- (2015) R. Frederick Ludlow et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Lessons from Hot Spot Analysis for Fragment-Based Drug Discovery
- (2015) David R. Hall et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- Efficient exploration of chemical space by fragment-based screening
- (2014) Richard J. Hall et al. PROGRESS IN BIOPHYSICS & MOLECULAR BIOLOGY
- Complementarity between in Silico and Biophysical Screening Approaches in Fragment-Based Lead Discovery against the A2A Adenosine Receptor
- (2013) Dan Chen et al. Journal of Chemical Information and Modeling
- Thermodynamics of Fragment Binding
- (2012) György G. Ferenczy et al. Journal of Chemical Information and Modeling
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