Journal
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Volume 58, Issue 18, Pages 6074-6078Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/anie.201900199
Keywords
alkaloids; natural products; oxidative coupling; regioselectivity; total synthesis
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Funding
- National Natural Science Foundation of China [21871013, 21572008]
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We report for the first time that the benzofuro[3,2-b]indoline framework could be obtained by PIDA-mediated direct oxidative coupling of 2,3-disubstituted-indoles with phenols. Application of this chemistry allows for an eight-step total synthesis of phalarine from commercially available tryptamine.
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