Silyl-Substituted Planar Chiral Phosphoric Acids with Ferrocene-bridged Paracyclophane Frameworks: Synthesis, Characterization, and Uses in Enantioselective aza-Friedel-Crafts Reactions

Stronger Brønsted Acids: Recent Progress

(2015) Takahiko Akiyama et al.   CHEMICAL REVIEWS

Strategies for the asymmetric functionalization of indoles: an update

(2015) Renato Dalpozzo   CHEMICAL SOCIETY REVIEWS

Recent Advances in Chiral Phosphoric Acid Catalyzed Asymmetric Reactions for the Synthesis of Enantiopure Indole Derivatives

(2015) Hua Wu et al.   SYNTHESIS-STUTTGART

Anticancer activity of VDR-coregulator inhibitor PS121912

(2014) Preetpal S. Sidhu et al.   CANCER CHEMOTHERAPY AND PHARMACOLOGY

Chiral Synthetic Equivalents of 2-Cyanoethyl Tetraisopropylphosphorodiamidite: Application to the Synthesis and Resolution of Chiral Phosphoric Acids

(2014) Kévin Isaac et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Planar Chiral Phosphoric Acids with Biphenylene-Tethered Paracyclophane Scaffolds: Synthesis, Characterization, and Catalytic Screening

(2014) Kévin Isaac et al.   JOURNAL OF ORGANIC CHEMISTRY

Development of Novel Vitamin D Receptor–Coactivator Inhibitors

(2014) Preetpal S. Sidhu et al.   ACS Medicinal Chemistry Letters

Development of Chiral Phosphoric Acids based on Ferrocene-Bridged Paracyclophane Frameworks

(2013) Jérémy Stemper et al.   ADVANCED SYNTHESIS & CATALYSIS

[3,3]Paracyclophanes as planar chiral scaffolds for the synthesis of new phosphoric acids

(2013) Jérémy Stemper et al.   CHEMICAL COMMUNICATIONS

Chiral Brønsted acid-catalyzed enantioselective ionic [2+4] cycloadditions

(2013) Alina Borovika et al.   TETRAHEDRON

Enantioselective Friedel–Crafts reactions between phenols and N-tosylaldimines catalyzed by a leucine-derived bifunctional catalyst

(2012) Guo-Xing Li et al.   CHEMICAL COMMUNICATIONS

Synthesis and application of the first planar chiral strong brønsted acid organocatalysts

(2012) Dieter Enders et al.   CHIRALITY

Discovery of the First Irreversible Small Molecule Inhibitors of the Interaction between the Vitamin D Receptor and Coactivators

(2012) Premchendar Nandhikonda et al.   JOURNAL OF MEDICINAL CHEMISTRY

Investigations of the marine flora and fauna of the Fiji Islands

(2012) Klaus-Dieter Feussner et al.   NATURAL PRODUCT REPORTS

Asymmetric spiroacetalization catalysed by confined Brønsted acids

(2012) Ilija Čorić et al.   NATURE

3-Substitued indoles: One-pot synthesis and evaluation of anticancer and Src kinase inhibitory activities

(2011) V. Kameshwara Rao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Chiral Brønsted acids in enantioselective carbonyl activations – activation modes and applications

(2011) Magnus Rueping et al.   CHEMICAL SOCIETY REVIEWS

Optically Active 1,1′-Spirobiindane-7,7′-diol (SPINOL)-Based Phosphoric Acids as Highly Enantioselective Catalysts for Asymmetric Organocatalysis

(2011) Chun-Hui Xing et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective Activation of Enantiotopic C(sp3)−Hydrogen by Means of Chiral Phosphoric Acid: Asymmetric Synthesis of Tetrahydroquinoline Derivatives

(2011) Keiji Mori et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Which Is the Actual Catalyst: Chiral Phosphoric Acid or Chiral Calcium Phosphate?

(2010) Manabu Hatano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A potent and selective indole N-type calcium channel (Cav2.2) blocker for the treatment of pain

(2010) Sriram Tyagarajan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A Useful Approach to Identify Novel Small-Molecule Inhibitors of Wnt-Dependent Transcription

(2010) K. Ewan et al.   CANCER RESEARCH

Organocatalytic strategies for the asymmetric functionalization of indoles

(2010) Giuseppe Bartoli et al.   CHEMICAL SOCIETY REVIEWS

Synthesis and Structural Aspects ofN-Triflylphosphoramides and Their Calcium Salts-Highly Acidic and Effective Brønsted Acids

(2010) Magnus Rueping et al.   CHEMISTRY-A EUROPEAN JOURNAL

Electron-Withdrawing, Biphenyl-2,2′-diol-Based Compounds for Asymmetric Catalysis

(2010) Elisa G. Gutierrez et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalyzed Asymmetric Friedel-Crafts Reactions

(2010) Vincent Terrasson et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

SPINOL-Derived Phosphoric Acids: Synthesis and Application in Enantioselective Friedel−Crafts Reaction of Indoles with Imines

(2010) Fangxi Xu et al.   JOURNAL OF ORGANIC CHEMISTRY

Kinetic Resolution of Homoaldols via Catalytic Asymmetric Transacetalization

(2010) Ilija Čorić et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Asymmetric Friedel-Crafts Reaction of 4,7-Dihydroindoles with Nitroolefins by Chiral Brønsted Acids under Low Catalyst Loading

(2009) Yi-Fei Sheng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective Synthesis of Fluorene Derivatives by Chiral Phosphoric Acid Catalyzed Tandem Double Friedel-Crafts Reaction

(2009) Feng-Lai Sun et al.   CHEMISTRY-A EUROPEAN JOURNAL

DFT Study on the Factors Determining the Enantioselectivity of Friedel−Crafts Reactions of Indole withN-Acyl andN-Tosylimines Catalyzed by BINOL−Phosphoric Acid Derivatives

(2009) Luis Simón et al.   JOURNAL OF ORGANIC CHEMISTRY

Chiral Phosphoric Acid Catalyzed Enantioselective Friedel–Crafts Alkylation of Indoles with Nitroalkenes: Cooperative Effect of 3 Å Molecular Sieves

(2008) Junji Itoh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Brønsted Acid Catalyzed Isoindoline Synthesis: Enhancement of Enantiomeric Ratio by Stereoablative Kinetic Resolution

(2008) Dieter Enders et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Development of Double Axially Chiral Phosphoric Acids and Their Catalytic Transfer Hydrogenation of Quinolines

(2008) Qun-Sheng Guo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Highly Enantioselective Friedel–Crafts Reaction of 4,7-Dihydroindoles with Imines by Chiral Phosphoric Acids: Facile Access to 2-Indolyl Methanamine Derivatives

(2008) Qiang Kang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Enantiopure (S)-Indolylglycine by Organocatalyzed Friedel–Crafts Alkylation of Indole

(2007) Martin J. Wanner et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY