Montelukast Disposition: No Indication of Transporter-Mediated Uptake in OATP2B1 and OATP1B1 Expressing HEK293 Cells

Assessment of absorption potential of poorly water-soluble drugs by using the dissolution/permeation system

(2013) Makoto Kataoka et al.   EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS

OATP1B1-related drug–drug and drug–gene interactions as potential risk factors for cerivastatin-induced rhabdomyolysis

(2013) Bani Tamraz et al.   Pharmacogenetics and Genomics

Classification of Inhibitors of Hepatic Organic Anion Transporting Polypeptides (OATPs): Influence of Protein Expression on Drug–Drug Interactions

(2012) Maria Karlgren et al.   JOURNAL OF MEDICINAL CHEMISTRY

Application of In Silico, In Vitro and Preclinical Pharmacokinetic Data for the Effective and Efficient Prediction of Human Pharmacokinetics

(2012) Kenneth H. Grime et al.   MOLECULAR PHARMACEUTICS

The Impact of Hepatic Uptake on the Pharmacokinetics of Organic Anions

(2011) P. Gardiner et al.   DRUG METABOLISM AND DISPOSITION

pH-Sensitive Interaction of HMG-CoA Reductase Inhibitors (Statins) with Organic Anion Transporting Polypeptide 2B1

(2011) Manthena V. Varma et al.   MOLECULAR PHARMACEUTICS

Comments on Mougey et al. (2009)

(2011) Xiaoyan Chu et al.   Pharmacogenetics and Genomics

Membrane transporters in drug development

(2010)   NATURE REVIEWS DRUG DISCOVERY

Interaction of HIV protease inhibitors with OATP1B1, 1B3, and 2B1

(2010) P. Annaert et al.   XENOBIOTICA

Montelukast in asthma: a review of its efficacy and place in therapy

(2010) Pierluigi Paggiaro et al.   Therapeutic Advances in Chronic Disease

Absorption of montelukast is transporter mediated: a common variant of OATP2B1 is associated with reduced plasma concentrations and poor response

(2009) Edward B. Mougey et al.   Pharmacogenetics and Genomics

Validation of cell-based OATP1B1 assays to assess drug transport and the potential for drug–drug interaction to support regulatory submissions

(2009) P. Sharma et al.   XENOBIOTICA

Dynamic Dissolution Testing To Establish In Vitro/In Vivo Correlations for Montelukast Sodium, a Poorly Soluble Drug

(2008) Arthur Okumu et al.   PHARMACEUTICAL RESEARCH