Engineering Cocrystals of Poorly Water-Soluble Drugs to Enhance Dissolution in Aqueous Medium
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Title
Engineering Cocrystals of Poorly Water-Soluble Drugs to Enhance Dissolution in Aqueous Medium
Authors
Keywords
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Journal
Pharmaceutics
Volume 10, Issue 3, Pages 108
Publisher
MDPI AG
Online
2018-08-01
DOI
10.3390/pharmaceutics10030108
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- Making Benzamide Cocrystals with Benzoic Acids: The Influence of Chemical Structure.
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- Solubility Advantage of Amorphous Drugs and Pharmaceutical Cocrystals
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- Hansen solubility parameter as a tool to predict cocrystal formation
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- Formulation design for poorly water-soluble drugs based on biopharmaceutics classification system: Basic approaches and practical applications
- (2011) Yohei Kawabata et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Cocrystallization and amorphization induced by drug–excipient interaction improves the physical properties of acyclovir
- (2011) Takaaki Masuda et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Solid forms of pharmaceuticals: Polymorphs, salts and cocrystals
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- Virtual cocrystal screening
- (2011) Daniele Musumeci et al. Chemical Science
- Application of Twin Screw Extrusion in the Manufacture of Cocrystals, Part I: Four Case Studies
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- Investigation of the Formation Process of Two Piracetam Cocrystals during Grinding
- (2011) Sönke Rehder et al. Pharmaceutics
- From unexpected reactions to a new family of ionic co-crystals: the case of barbituric acid with alkali bromides and caesium iodide
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- Cocrystal Eutectic Constants and Prediction of Solubility Behavior
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- Advantages of cocrystallization in the field of solid-state pharmaceutical chemistry: l-Proline and MnCl2
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- Ultrasound assisted cocrystallization from solution (USSC) containing a non-congruently soluble cocrystal component pair: Caffeine/maleic acid
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- New opportunities for materials synthesis using mechanochemistry
- (2010) Tomislav Friščić JOURNAL OF MATERIALS CHEMISTRY
- The Developability Classification System: Application of Biopharmaceutics Concepts to Formulation Development
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- Screening for pharmaceutical cocrystals using the supercritical fluid enhanced atomization process
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- Understanding and Predicting the Effect of Cocrystal Components and pH on Cocrystal Solubility
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- A Survey of Cocrystals Reported Prior to 2000
- (2009) G. Patrick Stahly CRYSTAL GROWTH & DESIGN
- Cambridge Structural Database Analysis of Molecular Complementarity in Cocrystals
- (2009) László Fábián CRYSTAL GROWTH & DESIGN
- Solubility Advantage of Pharmaceutical Cocrystals
- (2009) David J. Good et al. CRYSTAL GROWTH & DESIGN
- Synthesis and Structural Characterization of Cocrystals and Pharmaceutical Cocrystals: Mechanochemistry vs Slow Evaporation from Solution
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- Cocrystals of Caffeine and Hydroxybenzoic Acids Composed of Multiple Supramolecular Heterosynthons: Screening via Solution-Mediated Phase Transformation and Structural Characterization
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- Recent Advances in Understanding the Mechanism of Cocrystal Formation via Grinding
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- Pharmaceutical Cocrystals and Their Physicochemical Properties
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- Effects of Crystal Form on Solubility and Pharmacokinetics: A Crystal Engineering Case Study of Lamotrigine
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- Carbamazepine Co-crystallization with Pyridine Carboxamides: Rationalization by Complementary Phase Diagrams and Crystal Energy Landscapes
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- Dimorphs of a 1 : 1 cocrystal of ethenzamide and saccharin: solid-state grinding methods result in metastable polymorph
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- Formation of indomethacin–saccharin cocrystals using supercritical fluid technology
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- Can the Formation of Pharmaceutical Cocrystals Be Computationally Predicted? 2. Crystal Structure Prediction
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- Preparation and Characterization of Theophylline−Nicotinamide Cocrystal
- (2009) Jie Lu et al. ORGANIC PROCESS RESEARCH & DEVELOPMENT
- Polymorphs and Polymorphic Cocrystals of Temozolomide
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- Continuously Substituted Solid Solutions of Organic Co-Crystals
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- Co-Crystal Polymorphs from a Solvent-Mediated Transformation
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- Cocrystal Screening of Stanolone and Mestanolone Using Slurry Crystallization
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- Physicochemical Properties of Pharmaceutical Co-Crystals: A Case Study of Ten AMG 517 Co-Crystals
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- Hierarchy of Supramolecular Synthons: Persistent Carboxylic Acid···Pyridine Hydrogen Bonds in Cocrystals That also Contain a Hydroxyl Moiety
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- Polymorphism in Carbamazepine Cocrystals
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- Applying Hot-Stage Microscopy to Co-Crystal Screening: A Study of Nicotinamide with Seven Active Pharmaceutical Ingredients
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- Can the Formation of Pharmaceutical Cocrystals Be Computationally Predicted? I. Comparison of Lattice Energies
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- Cocrystals and Salts of Gabapentin: pH Dependent Cocrystal Stability and Solubility
- (2008) L. Sreenivas Reddy et al. CRYSTAL GROWTH & DESIGN
- Solid-State NMR Analysis of Organic Cocrystals and Complexes
- (2008) Frederick G. Vogt et al. CRYSTAL GROWTH & DESIGN
- Screening strategies based on solubility and solution composition generate pharmaceutically acceptable cocrystals of carbamazepine
- (2008) Scott L. Childs et al. CRYSTENGCOMM
- A rapid thermal method for cocrystal screening
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- Co-crystallisation of benzoic acid derivatives with N-containing bases in solution and by mechanical grinding: stoichiometric variants, polymorphism and twinning
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- Physical characterization and stability of amorphous indomethacin and ranitidine hydrochloride binary systems prepared by mechanical activation
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- Crystal engineering with acid and pyridine heteromeric synthon: neutral and ionic co-crystals
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- Isostructural polymorphs of triiodophloroglucinol and triiodoresorcinol
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- Ternary and quaternary co-crystals of 1,3-cis,5-cis-cyclohexanetricarboxylic acid and 4,4′-bipyridines
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