Possible sites of action of the new calcitonin gene-related peptide receptor antagonists

Effect of the calcitonin gene-related peptide (CGRP) receptor antagonist telcagepant in human cranial arteries

(2010) Lars Edvinsson et al.   CEPHALALGIA

Neurogenic inflammation: a study of rat trigeminal ganglion

(2010) Kim Anker Kristiansen et al.   JOURNAL OF HEADACHE AND PAIN

Characterization of the Calcitonin Gene-Related Peptide Receptor Antagonist Telcagepant (MK-0974) in Human Isolated Coronary Arteries

(2010) K. Y. Chan et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

New drugs in migraine treatment and prophylaxis: telcagepant and topiramate

(2010) Lars Edvinsson et al.   LANCET

Differential distribution of calcitonin gene-related peptide and its receptor components in the human trigeminal ganglion

(2010) S. Eftekhari et al.   NEUROSCIENCE

Calcitonin gene-related peptide differentially regulates gene and protein expression in trigeminal glia cells: Findings from array analysis

(2010) Carrie V. Vause et al.   NEUROSCIENCE LETTERS

CGRP receptor antagonism and migraine

(2010) Lars Edvinsson et al.   Neurotherapeutics

Brainstem and Thalamic Projections from a Craniovascular Sensory Nervous Centre in the Rostral Cervical Spinal Dorsal Horn of Rats

(2009) Y Liu et al.   CEPHALALGIA

Reduced Cerebellar Inhibition in Migraine with Aura: A TMS Study

(2009) Filippo Brighina et al.   CEREBELLUM

Effects of the prototype serotonin 5-HT1B/1D receptor agonist sumatriptan and the calcitonin gene-related peptide (CGRP) receptor antagonist CGRP8–37 on myocardial reactive hyperemic response in conscious dogs

(2009) Joseph J. Lynch et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Proinflammatory-Activated Trigeminal Satellite Cells Promote Neuronal Sensitization: Relevance for Migraine Pathology

(2009) Alessandro Capuano et al.   Molecular Pain

Randomized, controlled trial of telcagepant for the acute treatment of migraine

(2009) K. M. Connor et al.   NEUROLOGY

New insights in cerebellar function

(2009) P. Strata et al.   NEUROSCIENCE

Calcitonin gene-related peptide stimulation of nitric oxide synthesis and release from trigeminal ganglion glial cells

(2008) Jing Li et al.   BRAIN RESEARCH

The Blood-Brain Barrier in Migraine Treatment

(2008) L Edvinsson et al.   CEPHALALGIA

Calcitonin gene-related peptide (CGRP) triggers Ca2+responses in cultured astrocytes and in Bergmann glial cells from cerebellar slices

(2008) Stefano Morara et al.   EUROPEAN JOURNAL OF NEUROSCIENCE

Calcitonin receptor-like receptor (CLR), receptor activity-modifying protein 1 (RAMP1), and calcitonin gene-related peptide (CGRP) immunoreactivity in the rat trigeminovascular system: Differences between peripheral and central CGRP receptor distribution

(2008) Jochen K. Lennerz et al.   JOURNAL OF COMPARATIVE NEUROLOGY

Calcitonin Gene-Related Peptide Receptor Antagonism Does Not Affect the Severity of Myocardial Ischemia during Atrial Pacing in Dogs with Coronary Artery Stenosis

(2008) C. P. Regan et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Efficacy and tolerability of MK-0974 (telcagepant), a new oral antagonist of calcitonin gene-related peptide receptor, compared with zolmitriptan for acute migraine: a randomised, placebo-controlled, parallel-treatment trial

(2008) Tony W Ho et al.   LANCET

International Union of Pharmacology. LXIX. Status of the Calcitonin Gene-Related Peptide Subtype 2 Receptor

(2008) D. L. Hay et al.   PHARMACOLOGICAL REVIEWS