Synthesis and Evaluation of (S)-Proline-Containing α,β-Dipeptides as Organocatalysts in Solvent-Free Asymmetric Aldol Reactions Under Ball-Milling Conditions

Development of CN Coupling Using Mechanochemistry: Catalytic Coupling of Arylsulfonamides and Carbodiimides

(2014) Davin Tan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Corrigendum to “New class of bifunctional thioureas from l-proline: highly enantioselective Michael addition of 1,3-dicarbonyls to nitroolefins” [Tetrahedron: Asymmetry 25 (2014) 568–577]

(2014) Poopathy Vinayagam et al.   TETRAHEDRON-ASYMMETRY

New class of bifunctional thioureas from l-proline: highly enantioselective Michael addition of 1,3-dicarbonyls to nitroolefins

(2014) Poopathy Vinayagam et al.   TETRAHEDRON-ASYMMETRY

Design of Peptidyl Thiourea Derivatives as Organocatalysts for the Asymmetric Ring Opening ofmeso-Stilbene Oxides

(2014) Swapandeep Singh Chimni et al.   Asian Journal of Organic Chemistry

A Convenient Microwave-Assisted Propylphosphonic Anhydride (T3P®) Mediated One-Pot Pyrazolone Synthesis

(2013) Matthieu Desroses et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic solvent-free hydrogen bonding-mediated asymmetric Michael additions under ball milling conditions

(2013) Manuel Jörres et al.   GREEN CHEMISTRY

An Asymmetric Michael Addition of α,α-Disubstituted Aldehydes to Maleimides Leading to a One-Pot Enantioselective Synthesis of Lactones Catalyzed by Amino Acids

(2013) Christoforos G. Kokotos   ORGANIC LETTERS

Propanephosphonic Acid Anhydride (T3P®) - A Benign Reagent for Diverse Applications Inclusive of Large-Scale Synthesis

(2013) Vommina Sureshbabu et al.   SYNTHESIS-STUTTGART

β-tert-Butyl aspartate as an organocatalyst for the asymmetric α-amination of α,α-disubstituted aldehydes

(2013) Alexis Theodorou et al.   TETRAHEDRON

Higher enantioselectivities in thiourea-catalyzed Michael additions under solvent-free conditions

(2013) Martina Hestericová et al.   TETRAHEDRON

tert-Butyl esters of tripeptides based on Pro-Phe as organocatalysts for the asymmetric aldol reaction in aqueous or organic medium

(2013) Anastasia Psarra et al.   TETRAHEDRON

Mechanochemistry assisted asymmetric organocatalysis: A sustainable approach

(2012) Pankaj Chauhan et al.   Beilstein Journal of Organic Chemistry

Organocatalyst Efficiency in the Michael Additions of Aldehydes to Nitroalkenes in Water and in a Ball-Mill

(2012) Eva Veverková et al.   ChemCatChem

Recent efforts directed to the development of more sustainable asymmetric organocatalysis

(2012) José G. Hernández et al.   CHEMICAL COMMUNICATIONS

Click Mechanochemistry: Quantitative Synthesis of “Ready to Use” Chiral Organocatalysts by Efficient Two-Fold Thiourea Coupling to Vicinal Diamines

(2012) Vjekoslav Štrukil et al.   CHEMISTRY-A EUROPEAN JOURNAL

Preparation of Chiral Amino Esters by Asymmetric Phase-Transfer Catalyzed Alkylations of Schiff Bases in a Ball Mill

(2012) Pierrick Nun et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fast, solvent-free and hydrogen-bonding-mediated asymmetric Michael addition in a ball mill

(2012) Yi-Feng Wang et al.   GREEN CHEMISTRY

Synthesis of Versatile Bifunctional Derivatives of Chiral Diamines Obtained through Anchimerically Assisted Nucleophilic Substitution Reactions on Diastereomeric Phenylprolinols

(2012) Eusebio Juaristi et al.   HETEROCYCLES

Asymmetric Michael Additions of α-Nitrocyclohexanone to Aryl Nitroalkenes Catalyzed by Natural Amino Acid-Derived Bifunctional Thioureas

(2012) Manuel Jörres et al.   ORGANIC LETTERS

Multikilogram Synthesis of a Hepatoselective Glucokinase Activator

(2012) Joshua R. Dunetz et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

T3P (propylphosphonic anhydride) mediated conversion of Nα-protected amino/peptide acids into thioacids

(2012) Chilakapati Madhu et al.   TETRAHEDRON LETTERS

Asymmetric catalysis with peptides

(2011) Helma Wennemers   CHEMICAL COMMUNICATIONS

Asymmetric Aldol Reaction Organocatalyzed by (S)-Proline-Containing Dipeptides: Improved Stereoinduction under Solvent-Free Conditions

(2011) José G. Hernández et al.   JOURNAL OF ORGANIC CHEMISTRY

General and Scalable Amide Bond Formation with Epimerization-Prone Substrates Using T3P and Pyridine

(2011) Joshua R. Dunetz et al.   ORGANIC LETTERS

Recyclable Siloxy Serine Organocatalyst for the Direct Asymmetric Mannich Reactions in Ionic Liquids

(2011) Fui-Fong Yong et al.   SYNTHETIC COMMUNICATIONS

Efficient ball-mill procedure in the ‘green’ asymmetric aldol reaction organocatalyzed by (S)-proline-containing dipeptides in the presence of water

(2011) José G. Hernández et al.   TETRAHEDRON

Solvent-free asymmetric aldol reaction organocatalyzed by (S)-proline-containing thiodipeptides under ball-milling conditions

(2011) José G. Hernández et al.   TETRAHEDRON

Thiazolidine-based organocatalysts for a highly enantioselective direct aldol reaction

(2010) Raoní S. Rambo et al.   TETRAHEDRON-ASYMMETRY

A Novel Proline-Valinol Thioamide Small Organic Molecule for a Highly Enantioselective Direct Aldol Reaction

(2009) Bing Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of proline-derived dipeptides and their catalytic enantioselective direct aldol reactions: catalyst, solvent, additive and temperature effects

(2009) Y.-H. Chen et al.   AMINO ACIDS

Organocatalysis—after the gold rush

(2009) Søren Bertelsen et al.   CHEMICAL SOCIETY REVIEWS

Green Chemistry: Principles and Practice

(2009) Paul Anastas et al.   CHEMICAL SOCIETY REVIEWS

Proline−β3-Amino-Ester Dipeptides as Efficient Catalysts for Enantioselective Direct Aldol Reaction in Aqueous Medium

(2009) Mauro De Nisco et al.   JOURNAL OF ORGANIC CHEMISTRY

Development of a Practical Large-Scale Synthesis of Denagliptin Tosylate

(2009) Daniel E. Patterson et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Proline–threonine dipeptide as an organocatalyst for the direct asymmetric aldol reaction

(2009) Srivari Chandrasekhar et al.   TETRAHEDRON-ASYMMETRY

ProlinamidesversusProlinethioamides as Recyclable Catalysts in the Enantioselective Solvent-Free Inter- and Intramolecular Aldol Reactions

(2008) Diana Almaşi et al.   ADVANCED SYNTHESIS & CATALYSIS

New Simple Hydrophobic Proline Derivatives as Highly Active and Stereoselective Catalysts for the Direct Asymmetric Aldol Reaction in Aqueous Medium

(2008) Francesco Giacalone et al.   ADVANCED SYNTHESIS & CATALYSIS

Investigating Sequence Space: How Important is the Spatial Arrangement of Functional Groups in the Asymmetric Aldol Reaction Catalyst H-Pro-Pro-Asp-NH2?

(2008) Jefferson D. Revell et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly Diastereo- and Enantioselective Direct Aldol Reactions Promoted by Water-Compatible Organocatalysts Bearing Central and Axial Chiral Elements

(2008) Fang-Zhi Peng et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Aminocatalysis-Gold Rush in Organic Chemistry

(2008) Paolo Melchiorre et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Organocatalysis: From Infancy to Adolescence

(2008) Alessandro Dondoni et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Diastereo- and Enantioselective Direct Aldol Reaction Catalyzed by Simple Amphiphilic Proline Derivatives

(2008) Yu-Qin Fu et al.   CATALYSIS LETTERS

Hydrogen-Bond-Mediated Asymmetric Catalysis

(2008) Xinhong Yu et al.   Chemistry-An Asian Journal

Synthesis of Chiral Organocatalysts derived from Aziridines: Application in Asymmetric Aldol Reaction

(2008) Shikha Gandhi et al.   JOURNAL OF ORGANIC CHEMISTRY

A Highly Efficient Solvent-Free Asymmetric Direct Aldol Reaction Organocatalyzed by Recoverable (S)-Binam-l-Prolinamides. ESI-MS Evidence of the Enamine−Iminium Formation

(2008) Gabriela Guillena et al.   JOURNAL OF ORGANIC CHEMISTRY

Solid phase synthesis of novelα/β-tetrapeptides, electrospray ionization mass spectrometric evaluation of their metal cation complexation behavior, and conformational analysis using density functional theory (DFT)

(2008) Yamir Bandala et al.   JOURNAL OF PHYSICAL ORGANIC CHEMISTRY

Catalytic, Asymmetric Transannular Aldolizations: Total Synthesis of (+)-Hirsutene

(2008) Carley L. Chandler et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The advent and development of organocatalysis

(2008) David W. C. MacMillan   NATURE

Highly Enantioselective Aldol Reactions Catalyzed by a Recyclable Fluorous (S) Pyrrolidine Sulfonamide on Water

(2008) Liansuo Zu et al.   ORGANIC LETTERS

Synthesis of three novel chiral diamines derived from (S)-proline and their evaluation as precursors of diazaborolidines for the catalytic borane-mediated enantioselective reduction of prochiral ketones

(2008) J. Luis Olivares-Romero et al.   TETRAHEDRON

Sulfonamides of homoproline and dipeptides as organocatalysts for Michael and aldol reactions

(2008) Evaggelia Tsandi et al.   TETRAHEDRON

Toward an Artificial Aldolase

(2007) Daniel Font et al.   ORGANIC LETTERS