Total syntheses of indolactam alkaloids (−)-indolactam V, (−)-pendolmycin, (−)-lyngbyatoxin A, and (−)-teleocidin A-2

Enabling the Use of Heterocyclic Arynes in Chemical Synthesis

(2014) Adam E. Goetz et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of (−)-Epi-Indolactam V by an Intramolecular Buchwald–Hartwig C–N Coupling Cyclization Reaction

(2013) Michele Mari et al.   JOURNAL OF ORGANIC CHEMISTRY

Further Investigations into the Regioselectivity of 6,7-Indole Aryne Cyclo­additions with 2-Substituted Furans: Remarkable Contrasteric Preference Depends­ on Pyrrole and Benzene Ring Substitution

(2013) Keith Buszek et al.   SYNTHESIS-STUTTGART

Development of an Intramolecular Aryne Ene Reaction and Application to the Formal Synthesis of (±)-Crinine

(2012) David A. Candito et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total synthesis of (±)-cis-trikentrin B via intermolecular 6,7-indole aryne cycloaddition and Stille cross-coupling

(2012) Nalin Chandrasoma et al.   TETRAHEDRON LETTERS

Antimalarial β-Carboline and Indolactam Alkaloids from Marinactinospora thermotolerans, a Deep Sea Isolate

(2011) Hongbo Huang et al.   JOURNAL OF NATURAL PRODUCTS

Intramolecular Aryne–Ene Reaction: Synthetic and Mechanistic Studies

(2011) David A. Candito et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Overturning Indolyne Regioselectivities and Synthesis of Indolactam V

(2011) Sarah M. Bronner et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (−)-N-Methylwelwitindolinone C Isothiocyanate

(2011) Alexander D. Huters et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total synthesis of (−)-indolactam V

(2011) Zhengren Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Rh(I)-Catalyzed Ring-Opening of Hetaryne−Furan Diels−Alder Adducts: Rapid Access to Stereochemically Defined Heterocyclic Scaffolds

(2011) Trung D. Nguyen et al.   ORGANIC LETTERS

Application of 6,7-Indole Aryne Cycloaddition and Pd(0)-Catalyzed Suzuki–Miyaura and Buchwald–Hartwig Cross-Coupling Reactions for the Preparation of Annulated Indole Libraries

(2011) Paul D. Thornton et al.   ACS Combinatorial Science

Indolyne and Aryne Distortions and Nucleophilic Regioselectivites

(2010) Paul H.-Y. Cheong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indolyne Experimental and Computational Studies: Synthetic Applications and Origins of Selectivities of Nucleophilic Additions

(2010) G-Yoon J. Im et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

JBIR-31, a new teleocidin analog, produced by salt-requiring Streptomyces sp. NBRC 105896 isolated from a marine sponge

(2009) Miho Izumikawa et al.   JOURNAL OF ANTIBIOTICS

Synthesis and Evaluation of 3-Aroylindoles as Anticancer Agents: Metabolite Approach

(2009) Yu-Shan Wu et al.   JOURNAL OF MEDICINAL CHEMISTRY

A small molecule that directs differentiation of human ESCs into the pancreatic lineage

(2009) Shuibing Chen et al.   Nature Chemical Biology

Indolynes as Electrophilic Indole Surrogates: Fundamental Reactivity and Synthetic Applications

(2009) Sarah M. Bronner et al.   ORGANIC LETTERS

New synthesis of (±)-cis-trikentrin A via tandem indole aryne cycloaddition/Negishi reaction. Applications to library development

(2009) Neil Brown et al.   TETRAHEDRON LETTERS

Switchable Reactivity of Acylated α, β-Dehydroamino Ester in the Friedel−Crafts Alkylation of Indoles by Changing the Lewis Acid

(2008) Elena Angelini et al.   JOURNAL OF ORGANIC CHEMISTRY

Concise Total Synthesis of (±)-cis-Trikentrin A and (±)-Herbindole A via Intermolecular Indole Aryne Cycloaddition

(2008) Keith R. Buszek et al.   ORGANIC LETTERS

Regioselective Diels–Alder cycloadditions and other reactions of 4,5-, 5,6-, and 6,7-indole arynes

(2008) Neil Brown et al.   TETRAHEDRON LETTERS

Design and physicochemical properties of new fluorescent ligands of protein kinase C isozymes focused on CH/π interaction

(2007) Takuya Sugimoto et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, Conformational Analysis, and Biological Evaluation of 1-Hexylindolactam-V10 as a Selective Activator for Novel Protein Kinase C Isozymes

(2007) Ryo C. Yanagita et al.   JOURNAL OF MEDICINAL CHEMISTRY