Ligand-controlled β-selective C(sp3)–H arylation of N-Boc-piperidines

Synthesis of Aromatic α-Aminoesters: Palladium-Catalyzed Long-Range Arylation of Primary C sp 3H Bonds

(2012) Sam Aspin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

On the Mechanism of the Palladium-Catalyzed β-Arylation of Ester Enolates

(2012) Paolo Larini et al.   CHEMISTRY-A EUROPEAN JOURNAL

Direct α-Functionalization of Saturated Cyclic Amines

(2012) Emily A. Mitchell et al.   CHEMISTRY-A EUROPEAN JOURNAL

An Experimental and in Situ IR Spectroscopic Study of the Lithiation–Substitution of N-Boc-2-phenylpyrrolidine and -piperidine: Controlling the Formation of Quaternary Stereocenters

(2012) Nadeem S. Sheikh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transition metal-catalyzed arylation of unactivated C(sp3)–H bonds

(2011) Olivier Baudoin   CHEMICAL SOCIETY REVIEWS

Enantioselective, Palladium-Catalyzed α-Arylation ofN-Boc Pyrrolidine:In SituReact IR Spectroscopic Monitoring, Scope, and Synthetic Applications

(2011) Graeme Barker et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Diastereoselective Arylations of Substituted Piperidines

(2011) Stephanie Seel et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

sp3C–H Bond Activation with Ruthenium(II) Catalysts and C(3)-Alkylation of Cyclic Amines

(2011) Basker Sundararaju et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Development of a Fit-for-Purpose Large-Scale Synthesis of an Oral PARP Inhibitor

(2011) Debra J. Wallace et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Palladium-Catalyzed β Arylation of Carboxylic Esters

(2010) Alice Renaudat et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct Amination of Secondary Alcohols Using Ammonia

(2010) Dennis Pingen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Deprotonation ofN-Boc Piperidine: React IR Monitoring and Mechanistic Aspects

(2010) Darren Stead et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Application of Catalytic Dynamic Resolution ofN-Boc-2-lithiopiperidine to the Asymmetric Synthesis of 2-Aryl and 2-Vinyl Piperidines

(2010) Timothy K. Beng et al.   ORGANIC LETTERS

Dialkylbiaryl phosphines in Pd-catalyzed amination: a user's guide

(2010) David S. Surry et al.   Chemical Science

Biaryl Phosphane Ligands in Palladium-Catalyzed Amination

(2008) David S. Surry et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Practical Imidazole-Based Phosphine Ligands for Selective Palladium-Catalyzed Hydroxylation of Aryl Halides

(2008) Thomas Schulz et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 2-Arylpiperidines by Palladium Couplings of Aryl Bromides with Organozinc Species Derived from Deprotonation ofN-Boc-Piperidine

(2008) Iain Coldham et al.   ORGANIC LETTERS