Extending an In Vitro Panel for Estrogenicity Testing: The Added Value of Bioassays for Measuring Antiandrogenic Activities and Effects on Steroidogenesis

In vitro metabolism and bioavailability tests for endocrine active substances: What is needed next for regulatory purposes?

(2014) Miriam Jacobs   ALTEX-Alternatives to Animal Experimentation

A 155-plex high-throughput in vitro coregulator binding assay for (anti-)estrogenicity testing evaluated with 23 reference compounds

(2014) Si Wang   ALTEX-Alternatives to Animal Experimentation

Robust Array-Based Coregulator Binding Assay Predicting ERα-Agonist Potency and Generating Binding Profiles Reflecting Ligand Structure

(2013) Jac M. M. J. G. Aarts et al.   CHEMICAL RESEARCH IN TOXICOLOGY

History of oral contraceptive drugs and their use worldwide

(2012) Sophie Christin-Maitre   BEST PRACTICE & RESEARCH CLINICAL ENDOCRINOLOGY & METABOLISM

Screening for Modulatory Effects on Steroidogenesis Using the Human H295R Adrenocortical Cell Line: A Metabolomics Approach

(2012) Jeroen C. W. Rijk et al.   CHEMICAL RESEARCH IN TOXICOLOGY

Serine-305 Phosphorylation Modulates Estrogen Receptor Alpha Binding to a Coregulator Peptide Array, with Potential Application in Predicting Responses to Tamoxifen

(2012) R. Houtman et al.   MOLECULAR CANCER THERAPEUTICS

Structural and mechanistic insights into bisphenols action provide guidelines for risk assessment and discovery of bisphenol A substitutes

(2012) V. Delfosse et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Weak estrogenic transcriptional activities of Bisphenol A and Bisphenol S

(2012) Elise Grignard et al.   TOXICOLOGY IN VITRO

Selective Activation of Zebrafish Estrogen Receptor Subtypes by Chemicals by Using Stable Reporter Gene Assay Developed in a Zebrafish Liver Cell Line

(2011) Anne Cosnefroy et al.   TOXICOLOGICAL SCIENCES

The EDKB: an established knowledge base for endocrine disrupting chemicals

(2010) Don Ding et al.   BMC BIOINFORMATICS

Gynaecomastia linked to the intake of a herbal supplement fortified with diethylstilbestrol

(2010) A.W.F.T. Toorians et al.   Food Additives and Contaminants Part A-Chemistry Analysis Control Exposure & Risk Assessment

Superinduction of estrogen receptor mediated gene expression in luciferase based reporter gene assays is mediated by a post-transcriptional mechanism

(2010) A.M. Sotoca et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Computational Toxicology as Implemented by the U.S. EPA: Providing High Throughput Decision Support Tools for Screening and Assessing Chemical Exposure, Hazard and Risk

(2010) Robert Kavlock et al.   JOURNAL OF TOXICOLOGY AND ENVIRONMENTAL HEALTH-PART B-CRITICAL REVIEWS

Optimization and prevalidation of the in vitro ERα CALUX method to test estrogenic and antiestrogenic activity of compounds

(2010) Bart van der Burg et al.   REPRODUCTIVE TOXICOLOGY

Optimization and prevalidation of the in vitro AR CALUX method to test androgenic and antiandrogenic activity of compounds

(2010) Bart van der Burg et al.   REPRODUCTIVE TOXICOLOGY

In house validation of recombinant yeast estrogen and androgen receptor agonist and antagonist screening assays

(2010) S.N. Kolle et al.   TOXICOLOGY IN VITRO

SERMs and SARMs: Detection of their activities with yeast based bioassays

(2009) Toine F.H. Bovee et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Nuclear Receptor-Coregulator Interaction Profiling Identifies TRIP3 as a Novel Peroxisome Proliferator-activated Receptor γ Cofactor

(2009) Arjen Koppen et al.   MOLECULAR & CELLULAR PROTEOMICS

Inter-laboratory comparison of a yeast bioassay for the determination of estrogenic activity in biological samples

(2008) Toine F.H. Bovee et al.   ANALYTICA CHIMICA ACTA

Screening of synthetic and plant-derived compounds for (anti)estrogenic and (anti)androgenic activities

(2008) Toine F. H. Bovee et al.   ANALYTICAL AND BIOANALYTICAL CHEMISTRY