Deconstructive fluorination of cyclic amines by carbon-carbon cleavage

AgII -Mediated Synthesis of β-Fluoroketones by Oxidative Cyclopropanol Opening

(2017) Yuanlin Deng et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Selective Ring-Opening of N-Alkyl Pyrrolidines with Chloroformates to 4-Chlorobutyl Carbamates

(2017) Chunghyeon Yu et al.   JOURNAL OF ORGANIC CHEMISTRY

CF2H, a Hydrogen Bond Donor

(2017) Chanan D. Sessler et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Radical fluorination reactions by thermal and photoinduced methods

(2017) Beatriz Lantaño et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Late stage modification of peptides via C H activation reactions

(2017) Saumitra Sengupta et al.   TETRAHEDRON LETTERS

Silver-initiated radical ring expansion/fluorination of ethynyl cyclobutanols: efficient synthesis of monofluoroethenyl cyclopentanones

(2016) Qingshan Tian et al.   GREEN CHEMISTRY

Radicals: Reactive Intermediates with Translational Potential

(2016) Ming Yan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxidative diversification of amino acids and peptides by small-molecule iron catalysis

(2016) Thomas J. Osberger et al.   NATURE

Monofluorination of Organic Compounds: 10 Years of Innovation

(2015) Pier Alexandre Champagne et al.   CHEMICAL REVIEWS

Applications of Fluorine in Medicinal Chemistry

(2015) Eric P. Gillis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Mechanistic Study of Silver-Catalyzed Decarboxylative Fluorination

(2015) Niki R. Patel et al.   JOURNAL OF ORGANIC CHEMISTRY

Silver-Catalyzed Ring-Opening Strategy for the Synthesis of β- and γ-Fluorinated Ketones

(2015) Huijun Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A meta-selective C–H borylation directed by a secondary interaction between ligand and substrate

(2015) Yoichiro Kuninobu et al.   Nature Chemistry

Iron- or silver-catalyzed oxidative fluorination of cyclopropanols for the synthesis of β-fluoroketones

(2015) Shichao Ren et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Highly Chemoselective Aerobic Oxidation of Amino Alcohols into Amino Carbonyl Compounds

(2014) Yusuke Sasano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

N-Tosyl-(S)-Prolyl Chloride in Kinetic Resolution of Racemic Heterocyclic Amines

(2014) D. A. Gruzdev et al.   Chemistry of Heterocyclic Compounds

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

Direct, Catalytic Monofluorination of sp3 C–H Bonds: A Radical-Based Mechanism with Ionic Selectivity

(2014) Cody Ross Pitts et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Silver-Catalyzed Radical Fluorination of Alkylboronates in Aqueous Solution

(2014) Zhaodong Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Alkoxycarbonylpiperidines as N-nucleophiles in the palladium-catalyzed aminocarbonylation

(2014) Attila Takács et al.   MONATSHEFTE FUR CHEMIE

Straightforward synthesis of orthogonally protected piperidin-3-ylmethanamine and piperidin-4-ylmethanamine derivatives

(2014) Urban Košak et al.   TETRAHEDRON LETTERS

Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

(2013) Jiang Wang et al.   CHEMICAL REVIEWS

Future directions for peptide therapeutics development

(2013) Allan A. Kaspar et al.   DRUG DISCOVERY TODAY

Cesium Carbonate-Catalyzed Reduction of Amides with Hydrosilanes

(2013) Weilong Xie et al.   ORGANOMETALLICS

Tandem oxidative amidation of benzyl alcohols with amine hydrochloride salts catalysed by iron nitrate

(2013) Subhash Chandra Ghosh et al.   TETRAHEDRON LETTERS

Silver-Catalyzed Decarboxylative Fluorination of Aliphatic Carboxylic Acids in Aqueous Solution

(2012) Feng Yin et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis and evaluation of 18F labeled alanine derivatives as potential tumor imaging agents

(2012) Limin Wang et al.   NUCLEAR MEDICINE AND BIOLOGY

Copper-Catalyzed Direct Arylation of Cyclic Enamides Using Diaryliodonium Salts

(2012) Nicolas Gigant et al.   ORGANIC LETTERS

Construction of Nitrogen-Fused Tetrahydroquinolines via a Domino Reaction

(2012) Nicolas Gigant et al.   ORGANIC LETTERS

Synthesis and Conformational Analysis of Fluorinated Pipecolic Acids

(2012) Hamid Dhimane et al.   SYNLETT

Dehydrogenative amide synthesis from alcohol and amine catalyzed by hydrotalcite-supported gold nanoparticles

(2012) Jiangling Zhu et al.   TETRAHEDRON LETTERS

Green chemistry oriented organic synthesis in water

(2011) Marc-Olivier Simon et al.   CHEMICAL SOCIETY REVIEWS

Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

(2011) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

The Oxidation of Amides to Imides: A Powerful Synthetic Transformation

(2011) Jonathan Sperry   SYNTHESIS-STUTTGART

A New Highly Versatile Handle for Chemistry on a Solid Support: The Pipecolic Linker

(2010) Paweł Zajdel et al.   CHEMISTRY-A EUROPEAN JOURNAL

Bond Dissociation Energies of Solvated Silver(I)−Amide Complexes: Competitive Threshold Collision-Induced Dissociations and Calculations

(2010) Vladimir Romanov et al.   JOURNAL OF PHYSICAL CHEMISTRY A

Facile Procedure for Generating Side Chain Functionalized Poly(α-hydroxy acid) Copolymers from Aldehydes via a Versatile Passerini-Type Condensation

(2010) Mark Rubinshtein et al.   ORGANIC LETTERS

Ruthenium-Based Heterocyclic Carbene-Coordinated Olefin Metathesis Catalysts†

(2009) Georgios C. Vougioukalakis et al.   CHEMICAL REVIEWS

Synthetic therapeutic peptides: science and market

(2009) Patrick Vlieghe et al.   DRUG DISCOVERY TODAY

Synthesis and in Vitro and in Vivo Evaluation of18F-Labeled Positron Emission Tomography (PET) Ligands for Imaging the Vesicular Acetylcholine Transporter

(2009) Zhude Tu et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Two-Step, Formal [4 + 2] Approach toward Piperidin-4-ones via Au Catalysis

(2009) Li Cui et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Therapeutic application of peptides and proteins: parenteral forever?

(2009) Zuzana Antosova et al.   TRENDS IN BIOTECHNOLOGY

Binding Energies of the Silver Ion to Alcohols and Amides: A Theoretical and Experimental Study

(2008) Vladimir Romanov et al.   JOURNAL OF PHYSICAL CHEMISTRY A

Amidicity Change as a Significant Driving Force and Thermodynamic Selection Rule of Transamidation Reactions. A Synergy between Experiment and Theory

(2008) Zoltán Mucsi et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Ruthenium tetroxide oxidation of cyclic N-acylamines by a single layer method: formation of ω-amino acids

(2008) Mamoru Kaname et al.   TETRAHEDRON LETTERS

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS