Journal
ORGANIC LETTERS
Volume 11, Issue 23, Pages 5494-5496Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol9023453
Keywords
-
Categories
Funding
- Thailand Research Fund
- Center for Innovation in Chemistry (PERCH-CIC)
- Commission on Higher Education, Thai Ministry of Education
Ask authors/readers for more resources
Nucleophilic cleavage of enantiomerically pure 1,2-cyclic sulfamidates with phenol, aniline, and thiophenol nucleophiles, followed by a Mitsunobu reaction, including use of a o-quinomethide variant of this process, provides an entry to substituted 1,4-tetrahydrobenzoxazepines, benzothiazepines, and benzodiazepines. Application of this methodology to 1,3-cyclic sulfamidates affords a parallel entry to the analogous substituted 1,5-benzoxazocines and 1,5-benzodiazocines.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available