Journal
ORGANIC LETTERS
Volume 11, Issue 13, Pages 2788-2790Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol900943b
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Funding
- Chinese Academy of Sciences
- National Natural Science Foundation of China [20632050, 20621062]
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CuI-catalyzed coupling of 4-methylphenyl bromide with amino acids gives N-aryl amino acids, which are converted into linear dipeptides via iodination and condensation with L-Cysteine derived acyl chloride. Cyclization is achieved via a CuI/N,N-dimethylglycine catalyzed intramolecular coupling of aryl iodides with the liberated thiol to afford 1,5-benzothiazepine dipeptide mimetics.
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