Synthesis of (+)-L-733,060, (+)-CP-99,994 and (2S,3R)-3-hydroxypipecolic acid: Application of an organocatalytic direct vinylogous aldol reaction

The Vinylogous Aldol and Related Addition Reactions: Ten Years of Progress†

(2011) Giovanni Casiraghi et al.   CHEMICAL REVIEWS

A Stereoselective Route to cis-(2S,3R)-3-Hydroxypipecolic Acid and Two Enantiomeric cis-2-Hydroxymethyl-3-hydroxypiperidine Derivatives

(2011) Shital Chattopadhyay et al.   SYNTHESIS-STUTTGART

Asymmetric Direct Vinylogous Aldol Reaction of Furanone Derivatives Catalyzed by an Axially Chiral Guanidine Base

(2010) Hitoshi Ube et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic asymmetric direct vinylogous aldol reactions of γ-crotonolactone with aromatic aldehydes

(2010) Sunil V. Pansare et al.   CHEMICAL COMMUNICATIONS

Stereoselective Syntheses ofl-Pipecolic Acid and (2S,3S)-3-Hydroxypipecolic Acid from a ChiralN-Imino-2-phenyl-1,2-dihydropyridine Intermediate

(2010) Alexandre Lemire et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Direct Vinylogous Aldol Reaction of Unactivated γ-Butenolide to Aldehydes

(2010) Yang Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective α-Amination of 1,3-Dicarbonyl Compounds Using Squaramide Derivatives as Hydrogen Bonding Catalysts

(2010) Hideyuki Konishi et al.   ORGANIC LETTERS

Enantioselective Synthesis of (+)-l-733,060 and (+)-CP-99,994: Application of an Ireland-Claisen Rearrangement/Michael Addition Domino Sequence

(2010) Narciso Garrido et al.   SYNLETT

A stereoselective synthesis of (+)-L-733,060 from ethyl (R)-(+)-2,3-epoxypropanoate

(2010) Sébastien Prévost et al.   TETRAHEDRON-ASYMMETRY

Stereospecific, Flexible and Redox-Economic Asymmetric Synthesis ofcis- andtrans-3-Hydroxypipecolic Acids and ­Analogs

(2009) Bing Wang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of (+)-CP-99,994 via Pd(0)-Catalyzed Asymmetric Allylic and Homoallylic C−H Diamination of Terminal Olefin

(2009) Renzhong Fu et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalytic Asymmetric Synthesis of Piperidines from Pyrrolidine: Concise Synthesis of L-733,060§

(2009) Julia L. Bilke et al.   ORGANIC LETTERS

Asymmetric synthesis of (2S,3R)-(−)-epi-CP-99,994 using sulfinimine-derived anti-2,3-diamino esters

(2009) Franklin A. Davis et al.   TETRAHEDRON LETTERS

Synthesis of cis-3-hydroxypipecolic acid via SmI2-mediated cyclization of aldehydo β-aminovinyl sulfoxides

(2009) Hea Seung Chung et al.   TETRAHEDRON LETTERS

Synthesis of both enantiomers of hydroxypipecolic acid derivatives equivalent to 5-azapyranuronic acids and evaluation of their inhibitory activities against glycosidases

(2008) Yuichi Yoshimura et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Concise Asymmetric Synthesis of (+)-CP-99,994 and (+)-L-733,060 via Efficient Construction of Homochiralsyn-1,2-Diamines andsyn-1,2-Amino Alcohols

(2008) Run-Hua Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

A Convenient Access to the Piperidine Ring by Cyclization of Allylsilyl Substituted N- cyliminium and Iminium Ions: Application to the Synthesis of Piperidine Alkaloids.

(2008) R. Remuson et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

A Direct Stereoselective Approach totrans-2,3-Disubstituted Piperidines: Application in the Synthesis of 2-Epi-CP-99,994 and (+)-Epilupinine

(2008) M’hamed Ahari et al.   ORGANIC LETTERS

A short enantioselective synthesis of (+)-L-733,060 via Shi epoxidation of a homoallylic carboxylate

(2008) Lourdusamy Emmanuvel et al.   TETRAHEDRON LETTERS

Stereoselective total synthesis of (2S,3R)-3-hydroxypipecolic acid

(2008) Van-Thoai Pham et al.   TETRAHEDRON-ASYMMETRY

Recent advances in the stereoselective synthesis of trans-3,4-disubstituted-piperidines: applications to (−)-paroxetine

(2008) Carmela De Risi et al.   TETRAHEDRON-ASYMMETRY

Synthesis of pharmaceutically active compounds containing a disubstituted piperidine framework

(2007) Sara Källström et al.   BIOORGANIC & MEDICINAL CHEMISTRY

α-Amino 1,3-dithioketal mediated asymmetric synthesis of piperidines (L-733,060) and tetrahydrofuran glycines

(2007) Franklin A. Davis et al.   TETRAHEDRON LETTERS