Protecting-group-free synthesis of a dual CCK1/CCK2 receptor antagonist

Practical and Scalable Synthesis of a Selective CCK1Receptor Antagonist

(2010) Christopher M. Mapes et al.   JOURNAL OF ORGANIC CHEMISTRY

Anthranilic sulfonamide CCK1/CCK2 dual receptor antagonists II: Tuning of receptor selectivity and in vivo efficacy

(2009) Marna Pippel et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Anthranilic sulfonamide CCK1/CCK2 dual receptor antagonists I: Discovery of CCKR1 selectivity in a previously CCKR2-selective lead series

(2009) Marna Pippel et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The economies of synthesis

(2009) Timothy Newhouse et al.   CHEMICAL SOCIETY REVIEWS

Protecting-Group-Free Total Synthesis of (±)-Subincanadine F

(2009) Pinhong Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Protecting-group-free synthesis as an opportunity for invention

(2009) Ian S. Young et al.   Nature Chemistry

A Facile and Efficient Synthesis of 4-Hydroxy-2,6-cis-tetrahydropyrans via Tandem Cross-Metathesis/Thermal SN2′ Reaction: Protecting-Group-Free Synthesis of (±)-Diospongin A

(2009) Kiyoun Lee et al.   ORGANIC LETTERS

Protecting-Group-Free Synthesis of 3-tert-Prenylated Oxindoles: Contiguous All-Carbon Quaternary Centers via Tertiary Neopentyl Substitution

(2009) Christopher D. Grant et al.   ORGANIC LETTERS

A general method for the synthesis of benzimidazole-4-sulfonamides

(2009) Mark D. Rosen et al.   TETRAHEDRON LETTERS

An improved method of amide synthesis using acyl chlorides

(2009) Li Zhang et al.   TETRAHEDRON LETTERS

Discovery of potent cholecystokinin-2 receptor antagonists: Elucidation of key pharmacophore elements by X-ray crystallographic and NMR conformational analysis

(2008) Mark D. Rosen et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Tin triflate-mediated total synthesis of circumdatin F, sclerotigenin, asperlicin C, and other quinazolino[3,2-a][1,4]benzodiazepines

(2008) Ming-Chung Tseng et al.   CHEMICAL COMMUNICATIONS

A Protecting Group Free Synthesis of (±)-Neostenine via the [5 + 2] Photocycloaddition of Maleimides

(2008) Michael D. Lainchbury et al.   JOURNAL OF ORGANIC CHEMISTRY

Protecting Group Free Glycosidations Usingp-Toluenesulfonohydrazide Donors

(2008) Anna V. Gudmundsdottir et al.   ORGANIC LETTERS

Convenient synthesis of some optically active 1,4-benzodiazepin-2,5-diones

(2007) M. Bakavoli et al.   CHINESE CHEMICAL LETTERS

Synthesis and biological activities of a series of 4,5-diaryl-3-hydroxy-2(5H)-furanones

(2007) Fabrice Bailly et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY