Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 6, Issue 22, Pages 4093-4095Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/b816217b
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Funding
- EPSRC and sanofiaventis, Alnwick
- Engineering and Physical Sciences Research Council [GR/S90904/01] Funding Source: researchfish
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Syntheses of two 4-phenylpiperidines from bromobenzene have been developed involving anchoring to a fluorous-tag, Ir-catalysed borylation, Pd- and Co-catalysed elaboration then traceless cleavage. Although performed using 'cold' (i.e. unlabelled) bromobenzene as the starting material, these routes have been designed to minimise material loss via volatile intermediates and expedite purification during radiosynthesis from 'hot' (i.e. [C-14] labelled) bromobenzene.
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