Synthesis and Antiviral Evaluation of Novel 2′,2′-Difluoro 5′-Norcarbocyclic Phosphonic Acid Nucleosides as Antiviral Agents

Discovery of GS-9131: Design, synthesis and optimization of amidate prodrugs of the novel nucleoside phosphonate HIV reverse transcriptase (RT) inhibitor GS-9148

(2010) Richard L. Mackman et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Selective Ring-opening Fluorination of Epoxide: An Efficient Synthesis of 2'-C-Fluoro-2'-C-methyl Carbocyclic Nucleosides

(2010) Lian-Jin Liu et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Total synthesis of neomethymycin and novamethymycin

(2010) Hong-Se Oh et al.   TETRAHEDRON

Synthesis of branched 9-[2-(2-phosphonoethoxy)ethyl]purines as a new class of acyclic nucleoside phosphonates which inhibit Plasmodium falciparum hypoxanthine–guanine–xanthine phosphoribosyltransferase

(2009) Dana Hocková et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Recent advances in the synthesis of fluorinated nucleosides

(2009) Xiao-Long Qiu et al.   TETRAHEDRON

Synthesis and anti-HIV activity of GS-9148 (2′-Fd4AP), a novel nucleoside phosphonate HIV reverse transcriptase inhibitor

(2007) Constantine G. Boojamra et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS