Regioselective N-alkylation with alcohols for the preparation of 2-(N-alkylamino)quinazolines and 2-(N-alkylamino)pyrimidines

From Regioselective Condensation to Regioselective N-Alkylation: A Novel and Environmentally Benign Strategy for the Synthesis ofN,N′-Alkyl Aryl Ureas andN,N′-Dialkyl Ureas

(2013) Feng Li et al.   ChemCatChem

Iridium catalysed chemoselective alkylation of 2′-aminoacetophenone with primary benzyl type alcohols under microwave conditions

(2012) Shailen Bhat et al.   CHEMICAL COMMUNICATIONS

Highly Efficient Heterogeneous Gold-catalyzed Direct Synthesis of Tertiary and Secondary Amines from Alcohols and Urea

(2012) Lin He et al.   ChemSusChem

Regioselective N-Alkylation of 2-Aminoimidazoles with Alcohols to 2-(N-Alkylamino)imidazoles Catalyzed by the [Cp*IrCl2]2/K2CO3 System

(2012) Feng Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Mechanistic investigation of the iridium-catalysed alkylation of amines with alcohols

(2012) Peter Fristrup et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Selective Alkylation of (Hetero)Aromatic Amines with Alcohols Catalyzed by a Ruthenium Pincer Complex

(2012) Santosh Agrawal et al.   ORGANIC LETTERS

N-Alkylation of Amines with Alcohols Catalyzed by a Water-Soluble Cp*Iridium Complex: An Efficient Method for the Synthesis of Amines in Aqueous Media

(2011) Ryoko Kawahara et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of α-Amino Acid Amides: Ruthenium-Catalyzed Amination of α-Hydroxy Amides

(2011) Min Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Improved Ruthenium-Catalyzed Amination of Alcohols with Ammonia: Synthesis of Diamines and Amino Esters

(2011) Sebastian Imm et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Catalytic Amination of Alcohols

(2011) Sebastian Bähn et al.   ChemCatChem

Regioselective N-alkylation of 2-aminobenzothiazoles with benzylic alcohols

(2011) Feng Li et al.   CHEMICAL COMMUNICATIONS

Iridium-catalysed condensation of alcohols and amines as a method for aminosugar synthesis

(2011) Ian Cumpstey et al.   CHEMICAL COMMUNICATIONS

Direct N-alkylation of amino-azoles with alcohols catalyzed by an iridium complex/base system

(2011) Feng Li et al.   CHEMICAL COMMUNICATIONS

Organic Synthesis Involving Iridium-Catalyzed Oxidation

(2011) Takeyuki Suzuki   CHEMICAL REVIEWS

Pt-Sn/γ-Al2O3-Catalyzed Highly Efficient Direct Synthesis of Secondary and Tertiary Amines and Imines

(2011) Wei He et al.   CHEMISTRY-A EUROPEAN JOURNAL

Borrowing Hydrogen Methodology for Amine Synthesis under Solvent-Free Microwave Conditions

(2011) Andrew J. A. Watson et al.   JOURNAL OF ORGANIC CHEMISTRY

Impregnated Ruthenium on Magnetite as a Recyclable Catalyst for the N-Alkylation of Amines, Sulfonamides, Sulfinamides, and Nitroarenes Using Alcohols as Electrophiles by a Hydrogen Autotransfer Process

(2011) Rafael Cano et al.   JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Reductive Amination of Allylic Alcohols

(2011) Zeyneb Sahli et al.   ORGANIC LETTERS

Manganese Dioxide CatalyzedN-Alkylation of Sulfonamides and Amines with Alcohols under Air

(2011) Xiaochun Yu et al.   ORGANIC LETTERS

Use of an Iridium-Catalyzed Redox-Neutral Alcohol-Amine Coupling on Kilogram Scale for the Synthesis of a GlyT1 Inhibitor

(2011) Martin A. Berliner et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Organometallic hydrogen transfer and dehydrogenationcatalysts for the conversion of bio-renewable alcohols

(2011) Andrew C. Marr   Catalysis Science & Technology

Ruthenium-Catalyzed Cascade N- and C(3)-Dialkylation of Cyclic Amines with Alcohols Involving Hydrogen Autotransfer Processes

(2010) Basker Sundararaju et al.   ADVANCED SYNTHESIS & CATALYSIS

Amination of Aliphatic Alcohols and Diols with an Iridium Pincer Catalyst

(2010) Natalia Andrushko et al.   ChemCatChem

Iridium-catalysed amine alkylation with alcohols in water

(2010) Ourida Saidi et al.   CHEMICAL COMMUNICATIONS

New Iridium Catalysts for the Efficient Alkylation of Anilines by Alcohols under Mild Conditions

(2010) Stefan Michlik et al.   CHEMISTRY-A EUROPEAN JOURNAL

The “Borrowing Hydrogen Strategy” by Supported Ruthenium Hydroxide Catalysts: Synthetic Scope of Symmetrically and Unsymmetrically Substituted Amines

(2010) Kazuya Yamaguchi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Selective Ruthenium-Catalyzed N-Alkylation of Indoles by Using Alcohols

(2010) Sebastian Bähn et al.   CHEMISTRY-A EUROPEAN JOURNAL

Identification of Potent Pyrazolo[4,3-h]quinazoline-3-carboxamides as Multi-Cyclin-Dependent Kinase Inhibitors†

(2010) Gabriella Traquandi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia

(2010) Christopher D. Cox et al.   JOURNAL OF MEDICINAL CHEMISTRY

Swift and Efficient Synthesis of 4-Phenylquinazolines: Involvement ofN-Heterocyclic Carbene in the Key Cyclization Step

(2010) Julien Debray et al.   JOURNAL OF ORGANIC CHEMISTRY

Iridium- and ruthenium-catalysed synthesis of 2,3-disubstituted indoles from anilines and vicinal diols

(2010) Matyas Tursky et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Simple and Versatile Catalytic System for N-Alkylation of Sulfonamides with Various Alcohols

(2010) Mingwen Zhu et al.   ORGANIC LETTERS

Pd/C-catalyzed heterocyclization during copper-free Sonogashira coupling: synthesis of 2-benzylimidazo[1,2-a]pyrimidines in water

(2010) Mohammad Bakherad et al.   TETRAHEDRON LETTERS

Copper-Catalyzed Alkylation of Sulfonamides with Alcohols

(2009) Feng Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient Catalytic Synthesis of Tertiary and Secondary Amines from Alcohols and Urea

(2009) Jinling He et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-Pot Two-Step Solvent-Free Rapid and Clean Synthesis of 2-(Substituted Amino)pyrimidines by Microwave Irradiation

(2009) Shyamaprosad Goswami et al.   BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN

γ-Alumina-Supported Silver Cluster forN-Benzylation of Anilines with Alcohols

(2009) Kenichi Shimizu et al.   ChemCatChem

Hydrogen Autotransfer in theN-Alkylation of Amines and Related Compounds using Alcohols and Amines as Electrophiles

(2009) Gabriela Guillena et al.   CHEMICAL REVIEWS

Dehydrogenation as a Substrate-Activating Strategy in Homogeneous Transition-Metal Catalysis

(2009) Graham E. Dobereiner et al.   CHEMICAL REVIEWS

Selective Iridium-Catalyzed Alkylation of (Hetero)Aromatic Amines and Diamines with Alcohols under Mild Reaction Conditions

(2009) Benoît Blank et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ruthenium-catalyzed Selective Monoamination of Vicinal Diols

(2009) Sebastian Bähn et al.   ChemSusChem

Ruthenium-CatalyzedN-Alkylation of Amines and Sulfonamides Using Borrowing Hydrogen Methodology

(2009) M. Haniti S. A. Hamid et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Selective Synthesis of Primary Amines Directly from Alcohols and Ammonia

(2008) Chidambaram Gunanathan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

[IrCl2Cp*(NHC)] Complexes as Highly Versatile Efficient Catalysts for the Cross-Coupling of Alcohols and Amines

(2008) Amparo Prades et al.   CHEMISTRY-A EUROPEAN JOURNAL

Transition metal catalysed reactions of alcohols using borrowing hydrogen methodology

(2008) Tracy D. Nixon et al.   DALTON TRANSACTIONS

Synthesis of Copper Halide Coordination Polymers with Ligands Formed by In Situ Cyclization of 2-Aminopyrimidine and Ethanol

(2008) Minghui Bi et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Discovery of Highly Selective and Potent p38 Inhibitors Based on a Phthalazine Scaffold#

(2008) Brad Herberich et al.   JOURNAL OF MEDICINAL CHEMISTRY

Iridium and Ruthenium Complexes with Chelating N-Heterocyclic Carbenes: Efficient Catalysts for Transfer Hydrogenation, β-Alkylation of Alcohols, and N-Alkylation of Amines

(2008) Dinakar Gnanamgari et al.   ORGANOMETALLICS

Selective Synthesis of Secondary and Tertiary Amines by Cp*Iridium-Catalyzed Multialkylation of Ammonium Salts with Alcohols

(2007) Ryohei Yamaguchi et al.   ORGANIC LETTERS

Cp∗Ir-catalyzed N-alkylation of amines with alcohols. A versatile and atom economical method for the synthesis of amines

(2007) Ken-ichi Fujita et al.   TETRAHEDRON