A propofol binding site on mammalian GABAA receptors identified by photolabeling

A Single Phenylalanine Residue in the Main Intracellular Loop of α1 γ-Aminobutyric Acid Type A and Glycine Receptors Influences Their Sensitivity to Propofol

(2011) Gustavo Moraga-Cid et al.   ANESTHESIOLOGY

p-(4-Azipentyl)propofol: A Potent Photoreactive General Anesthetic Derivative of Propofol

(2011) Deirdre S. Stewart et al.   JOURNAL OF MEDICINAL CHEMISTRY

X-ray structures of general anaesthetics bound to a pentameric ligand-gated ion channel

(2011) Hugues Nury et al.   NATURE

Principles of activation and permeation in an anion-selective Cys-loop receptor

(2011) Ryan E. Hibbs et al.   NATURE

Numerous Classes of General Anesthetics Inhibit Etomidate Binding to γ-Aminobutyric Acid Type A (GABAA) Receptors

(2010) Guo-Dong Li et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

m-Azipropofol (AziPm) a Photoactive Analogue of the Intravenous General Anesthetic Propofol

(2010) Michael A. Hall et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Synthetic 18-Norsteroid Distinguishes between Two Neuroactive Steroid Binding Sites on GABAA Receptors

(2010) A. S. Evers et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

A Residue in Loop 9 of the β2-Subunit Stabilizes the Closed State of the GABAAReceptor

(2009) Carrie A. Williams et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Inverse Effects on Gating and Modulation Caused by a Mutation in the M2-M3 Linker of the GABAA Receptor   Subunit

(2009) S. M. O'Shea et al.   MOLECULAR PHARMACOLOGY

Gel-Based Mass Spectrometric Analysis of Recombinant GABAAReceptor Subunits Representing Strongly Hydrophobic Transmembrane Proteins

(2008) Sung Ung Kang et al.   JOURNAL OF PROTEOME RESEARCH

General anaesthesia: from molecular targets to neuronal pathways of sleep and arousal

(2008) Nicholas P. Franks   NATURE REVIEWS NEUROSCIENCE