Chelator-Accelerated One-Pot ‘Click’ Labeling of Small Molecule Tracers with 2-[18F]Fluoroethyl Azide

A One-Pot Three-Component Radiochemical Reaction for Rapid Assembly of 125I-Labeled Molecular Probes

(2012) Ran Yan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly efficient click labeling using 2-[18F]fluoroethyl azide and synthesis of an 18FN-hydroxysuccinimide ester as conjugation agent

(2012) Dong Zhou et al.   NUCLEAR MEDICINE AND BIOLOGY

Synthesis and evaluation of nucleoside radiotracers for imaging proliferation

(2012) Graham Smith et al.   NUCLEAR MEDICINE AND BIOLOGY

Radiolabelling and evaluation of novel haloethylsulfoxides as PET imaging agents for tumor hypoxia

(2012) Evelyn Laurens et al.   NUCLEAR MEDICINE AND BIOLOGY

Preparation of 18F-labeled peptides using the copper(I)-catalyzed azide-alkyne 1,3-dipolar cycloaddition

(2011) Herman S Gill et al.   Nature Protocols

‘Click labelling’ in PET radiochemistry

(2009) Matthias Glaser et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Recent Applications of Click Chemistry for the Synthesis of Radiotracers for Molecular Imaging

(2009) Constantin Mamat et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Methods for 18F-labeling of RGD peptides: comparison of aminooxy [18F]fluorobenzaldehyde condensation with ‘click labeling’ using 2-[18F]fluoroethylazide, and S-alkylation with [18F]fluoropropanethiol

(2008) Matthias Glaser et al.   AMINO ACIDS

Design, Synthesis, and Biological Characterization of a Caspase 3/7 Selective Isatin Labeled with 2-[18F]fluoroethylazide

(2008) Graham Smith et al.   JOURNAL OF MEDICINAL CHEMISTRY