{2-[1-(3-Methoxycarbonylmethyl-1H-indol-2-yl)-1-methyl-ethyl]-1H-indol-3-yl}-acetic acid methyl ester (MIAM): Its anti-cancer efficacy and intercalation mechanism identified via multi-model systems

Synthesis and structure–activity relationships of N-aryl(indol-3-yl)glyoxamides as antitumor agents

(2009) Pascal Marchand et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Potent antitumor bifunctional DNA alkylating agents, synthesis and biological activities of 3a-aza-cyclopenta[a]indenes

(2009) Rajesh Kakadiya et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII

(2009) Özlen Güzel et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

DNA-binding geometry dependent energy transfer from 4′,6-diamidino-2-phenylindole to cationic porphyrins

(2009) Biao Jin et al.   BIOPHYSICAL CHEMISTRY

Variolins and Related Alkaloids

(2009) Scott R. Walker et al.   CHEMICAL REVIEWS

Benzothiopyranoindole-Based Antiproliferative Agents: Synthesis, Cytotoxicity, Nucleic Acids Interaction, and Topoisomerases Inhibition Properties

(2009) Lisa Dalla Via et al.   JOURNAL OF MEDICINAL CHEMISTRY

Complex Network Spectral Moments for ATCUN Motif DNA Cleavage: First Predictive Study on Proteins of Human Pathogen Parasites

(2009) Cristian R. Munteanu et al.   JOURNAL OF PROTEOME RESEARCH

Synthesis, characterization, DNA-binding and DNA-photocleavage studies of [Ru(bpy)2(pmip)]2+ and [Ru(phen)2(pmip)]2+ (pmip=2-(2′-pyrimidyl)imidazo[4,5-f][1,10]phenanthroline

(2009) Shuo Shi et al.   POLYHEDRON

Indole-3-carbinol enhances anti-proliferative, but not anti-invasive effects of oxaliplatin in colorectal cancer cell lines

(2008) Lynne M. Howells et al.   BIOCHEMICAL PHARMACOLOGY

Synthesis of new heteroaryl and heteroannulated indoles from dehydrophenylalanines: Antitumor evaluation

(2008) Maria-João R.P. Queiroz et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and antitumor activity of novel enediyne-linked pyrrolo[2,1-c][1,4]benzodiazepine hybrids

(2008) Wan-Ping Hu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Induction of Apoptosis by DC-81-Indole Conjugate Agent Through NF-κB and JNK/AP-1 Pathway

(2008) Wan-Ping Hu et al.   CHEMICAL RESEARCH IN TOXICOLOGY

Synthesis and characterization of dinuclear macrocyclic cobalt(II), copper(II) and zinc(II) complexes derived from 2,2,2′,2′-S,S[bis(bis-N,N-2-thiobenzimidazolyloxalato-1,2-ethane)]: DNA binding and cleavage studies

(2008) Farukh Arjmand et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A novel indole ethyl isothiocyanate (7Me-IEITC) with anti-proliferative and pro-apoptotic effects on platinum-resistant human ovarian cancer cells

(2008) Rakesh K. Singh et al.   GYNECOLOGIC ONCOLOGY

Synthesis and Biological Evaluation of 1-Methyl-2-(3′,4′,5′-trimethoxybenzoyl)-3-aminoindoles as a New Class of Antimitotic Agents and Tubulin Inhibitors

(2008) Romeo Romagnoli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Identification, Characterization and Initial Hit-to-Lead Optimization of a Series of 4-Arylamino-3-Pyridinecarbonitrile as Protein Kinase C theta (PKCθ) Inhibitors

(2008) Derek C. Cole et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, DNA binding, and cytotoxicity of 1,4-bis(2-amino-ethylamino)anthraquinone–amino acid conjugates

(2007) Ling-Wei Hsin et al.   BIOORGANIC & MEDICINAL CHEMISTRY