A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds
Published 2015 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds
Authors
Keywords
-
Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 13, Issue 15, Pages 4570-4580
Publisher
Royal Society of Chemistry (RSC)
Online
2015-03-11
DOI
10.1039/c5ob00371g
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Synthesis of skeletally diverse alkaloid-like molecules: exploitation of metathesis substrates assembled from triplets of building blocks
- (2013) Sushil K Maurya et al. Beilstein Journal of Organic Chemistry
- A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling
- (2013) Henning S. G. Beckmann et al. Nature Chemistry
- Template-induced macrocycle diversity through large ring-forming alkylations of tryptophan
- (2013) Kenneth V. Lawson et al. TETRAHEDRON
- 2,5-Diketopiperazines: Synthesis, Reactions, Medicinal Chemistry, and Bioactive Natural Products
- (2012) Alan D. Borthwick CHEMICAL REVIEWS
- Grabbing for the Ring: Macrocycles Tweak the Conventions of Drug Making
- (2012) Wendy Wolfson CHEMISTRY & BIOLOGY
- Structure-Based Design of High-Affinity Macrocyclic Peptidomimetics to Block the Menin-Mixed Lineage Leukemia 1 (MLL1) Protein–Protein Interaction
- (2012) Haibin Zhou et al. JOURNAL OF MEDICINAL CHEMISTRY
- A diversity-oriented synthesis approach to macrocycles via oxidative ring expansion
- (2012) Felix Kopp et al. Nature Chemical Biology
- Protein–protein interaction inhibitors get into the groove
- (2012) Asher Mullard NATURE REVIEWS DRUG DISCOVERY
- A two-directional strategy for the diversity-oriented synthesis of macrocyclic scaffolds
- (2012) Kieron M. G. O'Connell et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Diverse organo-peptide macrocyclesvia a fast and catalyst-free oxime/intein-mediated dual ligation
- (2011) Maragani Satyanarayana et al. CHEMICAL COMMUNICATIONS
- Macrocycles Are Great Cycles: Applications, Opportunities, and Challenges of Synthetic Macrocycles in Drug Discovery
- (2011) Eric Marsault et al. JOURNAL OF MEDICINAL CHEMISTRY
- Contemporary strategies for peptide macrocyclization
- (2011) Christopher J. White et al. Nature Chemistry
- Diversity-oriented synthesis of macrocyclic peptidomimetics
- (2011) A. Isidro-Llobet et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Synthesis of Small Molecules with High Scaffold Diversity: Exploitation of Metathesis Cascades in Combination with Inter- and Intramolecular Diels-Alder Reactions
- (2010) Catherine O'Leary-Steele et al. CHEMISTRY-A EUROPEAN JOURNAL
- Expanding the range of ‘druggable’ targets with natural product-based libraries: an academic perspective
- (2010) Renato A Bauer et al. CURRENT OPINION IN CHEMICAL BIOLOGY
- “Clicktophycin-52”: A Bioactive Cryptophycin-52 Triazole Analogue
- (2010) Markus Nahrwold et al. ORGANIC LETTERS
- Diversity-oriented synthesis as a tool for the discovery of novel biologically active small molecules
- (2010) Warren R.J.D. Galloway et al. Nature Communications
- Probing the Bioactive Conformation of an Archetypal Natural Product HDAC Inhibitor with Conformationally Homogeneous Triazole-Modified Cyclic Tetrapeptides
- (2009) W. Seth Horne et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Total Synthesis of the Antibiotic Kendomycin by Macrocyclization using Photo-Fries Rearrangement and Ring-Closing Metathesis
- (2009) Thomas Magauer et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Synthesis and Antibacterial Activities ofN-Glycosylated Derivatives of Tyrocidine A, a Macrocyclic Peptide Antibiotic
- (2009) Honggang Hu et al. JOURNAL OF MEDICINAL CHEMISTRY
- Accessing Skeletal Diversity Using Catalyst Control: Formation ofnandn+ 1 Macrocyclic Triazole Rings
- (2009) Ann Rowley Kelly et al. ORGANIC LETTERS
- Synthesis of Natural-Product-Like Molecules with Over Eighty Distinct Scaffolds
- (2008) Daniel Morton et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Efficient parallel synthesis of macrocyclic peptidomimetics
- (2008) Eric Marsault et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Peptidomimetics, a synthetic tool of drug discovery
- (2008) Josef Vagner et al. CURRENT OPINION IN CHEMICAL BIOLOGY
- Multiple Multicomponent Macrocyclizations Including Bifunctional Building Blocks (MiBs) Based on Staudinger and Passerini Three-Component Reactions
- (2008) Fredy Leon et al. JOURNAL OF ORGANIC CHEMISTRY
- The exploration of macrocycles for drug discovery — an underexploited structural class
- (2008) Edward M. Driggers et al. NATURE REVIEWS DRUG DISCOVERY
- Diversity-oriented synthesis; a spectrum of approaches and results
- (2008) Richard J. Spandl et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Towards the Optimal Screening Collection: A Synthesis Strategy
- (2007) Thomas E. Nielsen et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreCreate your own webinar
Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.
Create Now