An improved procedure to prepare 3-methyl-4-nitroalkylenethylisoxazoles and their reaction under catalytic enantioselective Michael addition with nitromethane

Quality by design (QbD) of amide isosteres: 5,5-Disubstituted isoxazolines as potent CRTh2 antagonists with favorable pharmacokinetic and drug-like properties

(2014) Dong Xiao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Organocatalyzed asymmetric vinylogous Michael addition of α,β-unsaturated γ-butyrolactam

(2013) Jinlong Zhang et al.   CHEMICAL COMMUNICATIONS

The preparation of 3-methyl-4-nitro-5-(2-alkylethenyl)isoxazoles

(2013) Robert Wells et al.   TETRAHEDRON LETTERS

Trifluoromethylation of Aromatic Isoxazoles: Regio- and Diastereoselective Route to 5-Trifluoromethyl-2-isoxazolines

(2011) Hiroyuki Kawai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric 1,6-Michael Addition of Arylthiols to 3-Methyl-4-nitro-5-alkenyl-isoxazoles with Bifunctional Catalysts

(2011) Qing-Lan Pei et al.   JOURNAL OF ORGANIC CHEMISTRY

Studies on the reactivity of 3-methyl-4-nitro-5-styrylisoxazoles with S-nucleophiles

(2011) Simone Bruschi et al.   TETRAHEDRON LETTERS

Development of a Mild Procedure for the Addition of Bisulfite to Electrophilic Olefins

(2010) Francesco Fini et al.   ADVANCED SYNTHESIS & CATALYSIS

A Fast and Highly Efficient Protocol for Synthesis of Pyrrolo[2,3-d]isoxazoles and a New Series of Novel Benzyl Bis-pyrrolo[2,3-d]isoxazoles Using Task-Specific Ionic Liquids as Catalyst and Green Solvent

(2010) Eligeti Rajanarendar et al.   CHEMICAL & PHARMACEUTICAL BULLETIN

Preparation of mono-labelled aliphatic polyacids via isoxazole derivatives

(2010) Mauro F.A. Adamo et al.   TETRAHEDRON LETTERS

Catalytic Asymmetric Conjugate Addition of Nitroalkanes to 4-Nitro-5-styrylisoxazoles

(2009) Andrea Baschieri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A facile chemoenzymatic approach to chiral non-racemic β-alkyl-γ-amino acids and 2-alkylsuccinic acids. A concise synthesis of (S)-(+)-Pregabalin

(2008) Fulvia Felluga et al.   TETRAHEDRON-ASYMMETRY