Discovery, stereospecific characterization and peripheral modification of 1-(pyrrolidin-1-ylmethyl)-2-[(6-chloro-3-oxo-indan)-formyl]-1,2,3,4-tetrahydroisoquinolines as novel selective κ opioid receptor agonists

Synthesis of Tripeptides Containing d-Trp Substituted at the Indole Ring, Assessment of Opioid Receptor Binding and in Vivo Central Antinociception

(2014) Rossella De Marco et al.   JOURNAL OF MEDICINAL CHEMISTRY

Spinal and peripheral adenosine A1 receptors contribute to antinociception by tramadol in the formalin test in mice

(2013) Jana Sawynok et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Conformationally Constrained κ Receptor Agonists: Stereoselective Synthesis and Pharmacological Evaluation of 6,8-Diazabicyclo[3.2.2]nonane Derivatives†

(2010) Christian Geiger et al.   JOURNAL OF MEDICINAL CHEMISTRY

LPK-26, a novel κ-opioid receptor agonist with potent antinociceptive effects and low dependence potential

(2008) Yi-Min Tao et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Zonisamide Suppresses Pain Symptoms of Formalin-Induced Inflammatory and Streptozotocin-Induced Diabetic Neuropathy

(2008) Mitsuo Tanabe et al.   JOURNAL OF PHARMACOLOGICAL SCIENCES

Miniaturized Rotating Disk Intrinsic Dissolution Rate Measurement: Effects of Buffer Capacity in Comparisons to Traditional Wood’s Apparatus

(2008) Alex Avdeef et al.   PHARMACEUTICAL RESEARCH