Dual evaluation of some novel 2-amino-substituted coumarinylthiazoles as anti-inflammatory–antimicrobial agents and their docking studies with COX-1/COX-2 active sites

Pyridyl aminothiazoles as potent inhibitors of Chk1 with slow dissociation rates

(2012) Vadim Y. Dudkin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathway

(2012) Ian Bruce et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological activity of 2-aminothiazoles as novel inhibitors of PGE2 production in cells

(2012) Breland Smith et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Aminothiazoles as γ-secretase modulators

(2011) Thomas Lübbers et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Rofecoxib Analogues Possessing a Nitric Oxide Donor Sulfohydroxamic Acid (SO2NHOH) Cyclooxygenase-2 Pharmacophore: Synthesis, Molecular Modeling, and Biological Evaluation as Anti-inflammatory Agents

(2011) Atul Bhardwaj et al.   ChemMedChem

Synthesis and antimicrobial properties of some new thiazolyl coumarin derivatives

(2011) Afsheen Arshad et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2-Aminothiazoles as Therapeutic Leads for Prion Diseases

(2011) Alejandra Gallardo-Godoy et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of some pyrazole derivatives as anti-inflammatory–antibacterial agents

(2011) Pawan Kumar et al.   MEDICINAL CHEMISTRY RESEARCH

Synthesis, characterization and anti-microbial studies of some novel 2,4-disubstituted thiazoles

(2010) A.M. Vijesh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

High-throughput screening for inhibitors of Mycobacterium tuberculosis H37Rv

(2009) Subramaniam Ananthan et al.   TUBERCULOSIS

SAR and QSAR study on 2-aminothiazole derivatives, modulators of transcriptional repression in Huntington’s disease

(2008) Samantha Leone et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological activities of some new fluorinated coumarins and 1-aza coumarins

(2007) Rajesh G. Kalkhambkar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY