Steroid sulfatase inhibitors for estrogen- and androgen-dependent cancers

Aromatase and Dual Aromatase-Steroid Sulfatase Inhibitors from the Letrozole and Vorozole Templates

(2011) Paul M. Wood et al.   ChemMedChem

Effects of dehydroepiandrosterone on proliferation, migration, and death of breast cancer cells

(2011) Rebeca López-Marure et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Irosustat: a first-generation steroid sulfatase inhibitor in breast cancer

(2011) Carlo Palmieri et al.   Expert Review of Anticancer Therapy

Steroid sulfatase inhibitors: Promising new tools for breast cancer therapy?

(2011) Jürgen Geisler et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Development of steroid sulfatase inhibitors

(2011) L.W. Lawrence Woo et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Abiraterone and Increased Survival in Metastatic Prostate Cancer

(2011) Johann S. de Bono et al.   NEW ENGLAND JOURNAL OF MEDICINE

Increased estrogen sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1(17β-HSD1) following neoadjuvant aromatase inhibitor therapy in breast cancer patients

(2010) Niramol Chanplakorn et al.   BREAST CANCER RESEARCH AND TREATMENT

Preclinical pharmacokinetic, toxicological and biomarker evaluation of SR16157, a novel dual-acting steroid sulfatase inhibitor and selective estrogen receptor modulator

(2010) Linda Rausch et al.   CANCER CHEMOTHERAPY AND PHARMACOLOGY

Bicyclic Derivatives of the Potent Dual Aromatase-Steroid Sulfatase Inhibitor 2-Bromo-4-{[(4-cyanophenyl)(4H-1,2,4-triazol-4-yl)amino]methyl}phenylsulfamate: Synthesis, SAR, Crystal Structure, and in vitro and in vivo Activities

(2010) Paul M. Wood et al.   ChemMedChem

Steroid sulfatase and estrogen sulfotransferase in human carcinomas

(2010) Takashi Suzuki et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Environmental causes of cancer: endocrine disruptors as carcinogens

(2010) Ana M. Soto et al.   Nature Reviews Endocrinology

Partners in crime: deregulation of AR activity and androgen synthesis in prostate cancer

(2010) Karen E. Knudsen et al.   TRENDS IN ENDOCRINOLOGY AND METABOLISM

New Developments in Intracrinology of Human Breast Cancer

(2009) Hironobu Sasano et al.   Annals of the New York Academy of Sciences

A New Therapeutic Strategy against Hormone-Dependent Breast Cancer: The Preclinical Development of a Dual Aromatase and Sulfatase Inhibitor

(2008) P. A. Foster et al.   CLINICAL CANCER RESEARCH

The Use of Steroid Sulfatase Inhibitors as a Novel Therapeutic Strategy Against Hormone-Dependent Endometrial Cancer

(2008) Paul A. Foster et al.   ENDOCRINOLOGY

Estrone sulfatase activity in patients with advanced ovarian cancer

(2008) Justin C. Chura et al.   GYNECOLOGIC ONCOLOGY

Estrone sulfate (E1S), a prognosis marker for tumor aggressiveness in prostate cancer (PCa)

(2008) Frank Giton et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Inactivation of recombinant human steroid sulfatase by KW-2581

(2007) Hiroyuki Ishida et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY