Ligands Raise the Constraint That Limits Constitutive Activation in G Protein-coupled Opioid Receptors

Structure of the δ-opioid receptor bound to naltrindole

(2012) Sébastien Granier et al.   NATURE

Crystal structure of the µ-opioid receptor bound to a morphinan antagonist

(2012) Aashish Manglik et al.   NATURE

Ligand-Specific Interactions Modulate Kinetic, Energetic, and Mechanical Properties of the Human β2 Adrenergic Receptor

(2012) Michael Zocher et al.   STRUCTURE

Divergent agonist selectivity in activating β1- and β2-adrenoceptors for G-protein and arrestin coupling

(2011) Ida Casella et al.   BIOCHEMICAL JOURNAL

Crystal structure of the β2 adrenergic receptor–Gs protein complex

(2011) Søren G. F. Rasmussen et al.   NATURE

Morphine-like Opiates Selectively Antagonize Receptor-Arrestin Interactions

(2010) Paola Molinari et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Coupling of  2-Adrenoceptors to XL s and G s: A New Insight into Ligand-Induced G Protein Activation

(2009) A. I. Kaya et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Functional complementation of high-efficiency resonance energy transfer: a new tool for the study of protein binding interactions in living cells

(2007) Paola Molinari et al.   BIOCHEMICAL JOURNAL