A Competitive Inhibitor That Reduces Recruitment of Androgen Receptor to Androgen-responsive Genes

ARN-509: A Novel Antiandrogen for Prostate Cancer Treatment

(2012) N. J. Clegg et al.   CANCER RESEARCH

Androgen Receptor Exon 1 Mutation Causes Androgen Insensitivity by Creating Phosphorylation Site and Inhibiting Melanoma Antigen-A11 Activation of NH2- and Carboxyl-terminal Interaction-dependent Transactivation

(2012) William H. Lagarde et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Activation of the Androgen Receptor by Intratumoral Bioconversion of Androstanediol to Dihydrotestosterone in Prostate Cancer

(2011) James L. Mohler et al.   CANCER RESEARCH

Minireview: Alternative Activation Pathways for the Androgen Receptor in Prostate Cancer

(2011) Kristin R. Lamont et al.   MOLECULAR ENDOCRINOLOGY

Regression of Castrate-Recurrent Prostate Cancer by a Small-Molecule Inhibitor of the Amino-Terminus Domain of the Androgen Receptor

(2010) Raymond J. Andersen et al.   CANCER CELL

A Noncompetitive Small Molecule Inhibitor of Estrogen-regulated Gene Expression and Breast Cancer Cell Growth That Enhances Proteasome-dependent Degradation of Estrogen Receptor α

(2010) Nicole M. Kretzer et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Small Molecule Inhibitors as Probes for Estrogen and Androgen Receptor Action

(2010) David J. Shapiro et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Antitumour activity of MDV3100 in castration-resistant prostate cancer: a phase 1–2 study

(2010) Howard I Scher et al.   LANCET

Increased Expression of Androgen Receptor Coregulator MAGE-11 in Prostate Cancer by DNA Hypomethylation and Cyclic AMP

(2009) A. R. Karpf et al.   MOLECULAR CANCER RESEARCH

Inhibition of prostate cancer cell growth by second-site androgen receptor antagonists

(2009) J. D. Joseph et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Development of a Second-Generation Antiandrogen for Treatment of Advanced Prostate Cancer

(2009) C. Tran et al.   SCIENCE

A New Small Molecule Inhibitor of Estrogen Receptor α Binding to Estrogen Response Elements Blocks Estrogen-dependent Growth of Cancer Cells

(2008) Chengjian Mao et al.   JOURNAL OF BIOLOGICAL CHEMISTRY