Methylsulfonylnitrobenzoates, a New Class of Irreversible Inhibitors of the Interaction of the Thyroid Hormone Receptor and Its Obligate Coactivators That Functionally Antagonizes Thyroid Hormone

Molecular Aspects of Thyroid Hormone Actions

(2010) Sheue-Yann Cheng et al.   ENDOCRINE REVIEWS

Identification and Characterization of 4-Chloro-N-(2-{[5-trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide (GSK3787), a Selective and Irreversible Peroxisome Proliferator-Activated Receptor δ (PPARδ) Antagonist

(2010) Barry G. Shearer et al.   JOURNAL OF MEDICINAL CHEMISTRY

Novel Flufenamic Acid Analogues as Inhibitors of Androgen Receptor Mediated Transcription

(2009) Clémentine Féau et al.   ACS Chemical Biology

In VivoInteraction of Steroid Receptor Coactivator (SRC)-1 and the Activation Function-2 Domain of the Thyroid Hormone Receptor (TR) β in TRβ E457A Knock-In and SRC-1 Knockout mice

(2009) Manuela Alonso et al.   ENDOCRINOLOGY

Regulation of Pyruvate Dehydrogenase Kinase 4 (PDK4) by Thyroid Hormone

(2009) Ramy R. Attia et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Improvement of Pharmacological Properties of Irreversible Thyroid Receptor Coactivator Binding Inhibitors

(2009) Jong Yeon Hwang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Thyroid hormones and the control of cell proliferation or cell differentiation: Paradox or duality?

(2009) Elsa Kress et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Nuclear receptor drug discovery

(2008) Taosheng Chen   CURRENT OPINION IN CHEMICAL BIOLOGY

Implications of the binding of tamoxifen to the coactivator recognition site of the estrogen receptor

(2008) D. J Kojetin et al.   ENDOCRINE-RELATED CANCER

Structural and Biochemical Basis for the Binding Selectivity of Peroxisome Proliferator-activated Receptor γ to PGC-1α

(2008) Yong Li et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Blocking Estrogen Signaling After the Hormone: Pyrimidine-Core Inhibitors of Estrogen Receptor-Coactivator Binding

(2008) Alexander A. Parent et al.   JOURNAL OF MEDICINAL CHEMISTRY

Comprehensive Mechanistic Analysis of Hits from High-Throughput and Docking Screens against β-Lactamase

(2008) Kerim Babaoglu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Ligand induced interaction of thyroid hormone receptor beta with its coregulators

(2008) Napoleão F. Valadares et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Complex actions of thyroid hormone receptor antagonist NH-3 on gene promoters in different cell lines

(2008) Vanya Shah et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Access and Binding of Local Anesthetics in the Closed Sodium Channel

(2008) I. Bruhova et al.   MOLECULAR PHARMACOLOGY

Tamoxifen (ICI46,474) as a targeted therapy to treat and prevent breast cancer

(2006) V Craig Jordan   BRITISH JOURNAL OF PHARMACOLOGY